Compile Data Set for Download or QSAR
Report error Found 148 Enz. Inhib. hit(s) with all data for entry = 50028725
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250081([Hyp2]PACAP38 | CHEMBL499507)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250076([Nal6]PACAP27 | CHEMBL525613)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250033([Ala7]PACAP38 | CHEMBL525419)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250074([Bip6]PACAP27 | CHEMBL507480)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250075([Bip6]PACAP38 | CHEMBL526315)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250077([Nal6]PACAP38 | CHEMBL503123)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250069([Glu3]PACAP38 | CHEMBL524494)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250019(PACAP | PACAP-38 | CHEMBL524658 | PACAP(1-38) | PA...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250080([Hyp2]PACAP27 | CHEMBL524495)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250061([His(1-Me)1]PACAP38 | CHEMBL498948)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250071([Cha6]PACAP38 | CHEMBL524683)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250073([Tyr6]PACAP38 | CHEMBL526360)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250035([D-His1]PACAP38 | CHEMBL525073)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250087([Aib4]PACAP38 | CHEMBL499665)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250033([Ala7]PACAP38 | CHEMBL525419)
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250037([D-Ser2]PACAP38 | CHEMBL524894)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250079([Pro2]PACAP38 | CHEMBL506840)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250085([Aib2]PACAP38 | CHEMBL506517)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250059(Ac-PACAP38 | CHEMBL530563)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250074([Bip6]PACAP27 | CHEMBL507480)
Affinity DataIC50: 4.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250034([D-His1]PACAP27 | CHEMBL499781)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250077([Nal6]PACAP38 | CHEMBL503123)
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250023(CHEMBL500280 | [Ala2]PACAP(1-38) | [Ala2]PACAP38)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250022([Ala2]PACAP27 | CHEMBL525392)
Affinity DataIC50: 5.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250035([D-His1]PACAP38 | CHEMBL525073)
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250075([Bip6]PACAP38 | CHEMBL526315)
Affinity DataIC50: 5.40nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250018(PACAP27 | CHEMBL524852)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250059(Ac-PACAP38 | CHEMBL530563)
Affinity DataIC50: 5.70nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250019(PACAP | PACAP-38 | CHEMBL524658 | PACAP(1-38) | PA...)
Affinity DataIC50: 6.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250076([Nal6]PACAP27 | CHEMBL525613)
Affinity DataIC50: 6.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250037([D-Ser2]PACAP38 | CHEMBL524894)
Affinity DataIC50: 6.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250071([Cha6]PACAP38 | CHEMBL524683)
Affinity DataIC50: 6.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250073([Tyr6]PACAP38 | CHEMBL526360)
Affinity DataIC50: 6.70nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250022([Ala2]PACAP27 | CHEMBL525392)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250069([Glu3]PACAP38 | CHEMBL524494)
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250085([Aib2]PACAP38 | CHEMBL506517)
Affinity DataIC50: 7.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250039([D-Asp3]PACAP38 | CHEMBL524334)
Affinity DataIC50: 7.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250036([D-Ser2]PACAP27 | CHEMBL506133)
Affinity DataIC50: 7.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250045([D-Thr7]PACAP38 | CHEMBL525230)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250027([Ala4]PACAP38 | CHEMBL525091)
Affinity DataEC50:  7.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250078([Pro2]PACAP27 | CHEMBL524672)
Affinity DataEC50:  7.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250061([His(1-Me)1]PACAP38 | CHEMBL498948)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250039([D-Asp3]PACAP38 | CHEMBL524334)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250072([Tyr6]PACAP27 | CHEMBL498867)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250078([Pro2]PACAP27 | CHEMBL524672)
Affinity DataIC50: 7.80nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250023(CHEMBL500280 | [Ala2]PACAP(1-38) | [Ala2]PACAP38)
Affinity DataIC50: 7.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250072([Tyr6]PACAP27 | CHEMBL498867)
Affinity DataIC50: 7.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250058(Ac-PACAP27 | CHEMBL505046)
Affinity DataIC50: 8.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250018(PACAP27 | CHEMBL524852)
Affinity DataIC50: 8.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250036([D-Ser2]PACAP27 | CHEMBL506133)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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