Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50033463
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345895BDBM50345895(1-((3-amino-6-cyclopropylpyrazin-2-yl)methyl)-3-(2...)
Affinity DataIC50: 15nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345893BDBM50345893(1-((3-amino-6-propylpyrazin-2-yl)methyl)-3-(2-oxo-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345894BDBM50345894(1-((3-amino-6-butylpyrazin-2-yl)methyl)-3-(2-oxo-2...)
Affinity DataIC50: 30nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345891BDBM50345891(tert-butyl 4-(3-((3-amino-6-propylpyrazin-2-yl)met...)
Affinity DataIC50: 45nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345896BDBM50345896(1-(4-(3-((3-amino-6-cyclopropylpyrazin-2-yl)methyl...)
Affinity DataIC50: 83nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345892BDBM50345892(tert-butyl 4-(3-((3-amino-6-cyclopropylpyrazin-2-y...)
Affinity DataIC50: 103nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345890BDBM50345890(tert-butyl 4-(3-((3-amino-6-ethylpyrazin-2-yl)meth...)
Affinity DataIC50: 140nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345870BDBM50345870(isobutyl 4-(3-((3-amino-6-chloropyrazin-2-yl)methy...)
Affinity DataIC50: 150nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345871BDBM50345871(tert-butyl 4-(3-((3-amino-6-chloropyrazin-2-yl)met...)
Affinity DataIC50: 190nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345875BDBM50345875(tert-butyl 4-(3-((3-amino-6-methylpyrazin-2-yl)met...)
Affinity DataIC50: 210nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345884BDBM50345884(1-((3-amino-6-methylpyrazin-2-yl)methyl)-3-(2-oxo-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345869BDBM50345869(butyl 4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)t...)
Affinity DataIC50: 230nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345868BDBM50345868(ethyl 4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)t...)
Affinity DataIC50: 310nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345852BDBM50345852(benzyl 4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)...)
Affinity DataIC50: 460nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345832BDBM50345832(1-((3-amino-6-cyclopropylpyrazin-2-yl)methyl)-3-ph...)
Affinity DataIC50: 470nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345883BDBM50345883(N-(4-(3-((3-amino-6-methylpyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 580nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345874BDBM50345874(1-(4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 700nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345876BDBM50345876(phenyl 4-(3-((3-amino-6-methylpyrazin-2-yl)methyl)...)
Affinity DataIC50: 730nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345867BDBM50345867(methyl 4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)...)
Affinity DataIC50: 940nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345854BDBM50345854(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(2-chlo...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345881BDBM50345881(N-(4-(3-((3-amino-6-methylpyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345829BDBM50345829(1-((3-amino-6-ethylpyrazin-2-yl)methyl)-3-phenylth...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345872BDBM50345872(isobutyl 4-(3-((3-amino-6-chloropyrazin-2-yl)methy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345873BDBM50345873(1-(4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345839BDBM50345839(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-meth...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345814BDBM50345814(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-phenylt...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345856BDBM50345856(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(2-fluo...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345851BDBM50345851(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-amin...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345830BDBM50345830(1-((3-amino-6-propylpyrazin-2-yl)methyl)-3-phenylt...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345880BDBM50345880(N-(4-(3-((3-amino-6-methylpyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345862BDBM50345862(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(2,4-di...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345817BDBM50345817(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-tert-bu...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345857BDBM50345857(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(2-(met...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345855BDBM50345855(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(2-meth...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345840BDBM50345840(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-isop...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345846BDBM50345846(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-(ben...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345837BDBM50345837(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-p-tolyl...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345878BDBM50345878(4-(3-((3-amino-6-methylpyrazin-2-yl)methyl)thioure...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345842BDBM50345842(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-brom...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345826BDBM50345826(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(naphth...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345853BDBM50345853(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-o-tolyl...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345838BDBM50345838(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-chlo...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345882BDBM50345882(N-(4-(3-((3-amino-6-methylpyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345828BDBM50345828(1-((3-amino-6-methylpyrazin-2-yl)methyl)-3-phenylt...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345863BDBM50345863(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(2,4-di...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345850BDBM50345850(N-(4-(3-((3-amino-6-chloropyrazin-2-yl)methyl)thio...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345847BDBM50345847(1-(4-acetylphenyl)-3-((3-amino-6-chloropyrazin-2-y...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345844BDBM50345844(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-cyan...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345849BDBM50345849(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-(4-(dim...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345859BDBM50345859(1-((3-amino-6-chloropyrazin-2-yl)methyl)-3-m-tolyl...)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of MK2 using biotin-LCAYSRALSRQLSSGVSEIRH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
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