Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50028826
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268430((S)-N-((S)-1-amino-3-(3-tert-butyl-4-hydroxyphenyl...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268433((S)-2-((S)-2-amino-N-methyl-3-phenylpropanamido)-N...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268432((S)-N-((S)-1-amino-3-(3-tert-butyl-4-hydroxyphenyl...)
Affinity DataIC50:  4.30nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268377((S)-2-amino-N-((S)-1-((S)-1-amino-3-(3-tert-butyl-...)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268378((S)-2-amino-N-((3S,6S)-3-(3-tert-butyl-4-hydroxybe...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268376((S)-2-amino-N-((S)-2-((S)-1-amino-3-(3-tert-butyl-...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268431((S)-N-((S)-1-amino-3-(3-tert-butyl-4-hydroxyphenyl...)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268429((S)-N-((S)-1-amino-3-(3-tert-butyl-4-hydroxyphenyl...)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268428((S)-N-((S)-1-amino-3-(3-tert-butyl-4-hydroxyphenyl...)
Affinity DataIC50:  46nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Oryctolagus cuniculus)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268427((S)-2-amino-N-((S)-1-((S)-1-amino-3-(3-tert-butyl-...)
Affinity DataIC50:  185nMAssay Description:Displacement of [125I]motilin from MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed