Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50038925
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as increase in intracellular calcium release by fluorescence assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataIC50: 1.51E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378134(CHEMBL572657)
Affinity DataIC50: 9.20E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378133(CHEMBL584184)
Affinity DataIC50: 1.66E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378128(CHEMBL575653)
Affinity DataIC50: 2.64E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378126(CHEMBL572422)
Affinity DataIC50: 2.67E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378130(CHEMBL574076)
Affinity DataIC50: 3.38E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378124(CHEMBL572897)
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378127(CHEMBL574998)
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378129(CHEMBL575649)
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378131(CHEMBL575202)
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378132(CHEMBL574529)
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378123(CHEMBL582936)
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378125(CHEMBL572655)
Affinity DataIC50: 5.96E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 3 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed