Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50030441
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296238((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296237((2R,3R)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296238((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296239((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296235((-)-Epigallocatechin-3-(4''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296236((2R,3R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296235((-)-Epigallocatechin-3-(4''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296239((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296238((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296241((2R,3S)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296240((2R,3S)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296239((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296237((2R,3R)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296240((2R,3S)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296235((-)-Epigallocatechin-3-(4''-O-methyl)gallate | (2R...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296236((2R,3R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296241((2R,3S)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296240((2R,3S)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296236((2R,3R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296237((2R,3R)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296241((2R,3S)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed