Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50000825 Sort by
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010272(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010273(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  100nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010271(CHEMBL111425 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  800nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010274(CHEMBL328561 | Acetic acid (3R,4aR,5S,6S,6aS,10S,1...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010266(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  82nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010273(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  53nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010270(CHEMBL111514 | Acetic acid 6-[2-(2-bromo-acetylami...)
Affinity DataKd:  1.70E+4nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010274(CHEMBL328561 | Acetic acid (3R,4aR,5S,6S,6aS,10S,1...)
Affinity DataKd:  34nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010260(CHEMBL107566 | [2-(2-Bromo-acetylamino)-ethyl]-car...)
Affinity DataKd:  1.30E+3nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010271(CHEMBL111425 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  60nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010265(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  13nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010275(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010269(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Affinity DataKd:  240nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010275(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  174nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010262(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  80nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010268(CHEMBL91909 | (2-Amino-ethyl)-carbamic acid (3R,4a...)
Affinity DataKd:  98nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010261(colforsinum | cid_47936 | colforsina | colforsine ...)
Affinity DataKd:  29nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010266(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  400nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010260(CHEMBL107566 | [2-(2-Bromo-acetylamino)-ethyl]-car...)
Affinity DataKd:  10nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010261(colforsinum | cid_47936 | colforsina | colforsine ...)
Affinity DataKd:  5.00E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010263(CHEMBL107985 | Acetic acid 10,10b-dihydroxy-6-(2-i...)
Affinity DataKd:  300nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010262(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010264(CHEMBL110686 | (2-Isothiocyanato-ethyl)-carbamic a...)
Affinity DataKd:  110nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010259(CHEMBL326463 | Acetic acid 10,10b-dihydroxy-6-{2-[...)
Affinity DataKd:  9nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010263(CHEMBL107985 | Acetic acid 10,10b-dihydroxy-6-(2-i...)
Affinity DataKd:  130nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010265(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  1.10E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010259(CHEMBL326463 | Acetic acid 10,10b-dihydroxy-6-{2-[...)
Affinity DataKd:  2.80E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010267([2-(4-Hydroxy-phenyl)-ethyl]-carbamic acid (3R,4aR...)
Affinity DataKd:  236nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010267([2-(4-Hydroxy-phenyl)-ethyl]-carbamic acid (3R,4aR...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010268(CHEMBL91909 | (2-Amino-ethyl)-carbamic acid (3R,4a...)
Affinity DataKd:  2.80E+4nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010269(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Affinity DataKd:  61nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010264(CHEMBL110686 | (2-Isothiocyanato-ethyl)-carbamic a...)
Affinity DataKd:  500nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010270(CHEMBL111514 | Acetic acid 6-[2-(2-bromo-acetylami...)
Affinity DataKd:  10nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenylate cyclase type 1(Bovine)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010272(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  94nMAssay Description:Displacement of [125I]6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed