Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50030377
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295298(CHEMBL552717 | icterogenin regioisomer)
Affinity DataKi:  5.30E+3nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295299(1-O-[alpha-L-(Rhamnopyranosyl]-23-acetoxy-3beta-ac...)
Affinity DataKi:  7.20E+3nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295300(CHEMBL554122 | icterogenin)
Affinity DataKi:  7.60E+3nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295301(23-O-[alpha-L-(2',4'-Diacetylrhamnopyranosyl]imber...)
Affinity DataKi:  1.41E+4nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295302(23-acetoxy-3beta-acetylimberbic acid | CHEMBL53990...)
Affinity DataKi:  1.78E+4nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295308(1-O-[alpha-L-(Rhamnopyranosyl]-23-acetoxy-3beta-ac...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295309(23-O-[alpha-L-(4'-Acetylrhamnopyranosyl]-3beta-ace...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295310(CHEMBL540988 | lantadene A)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295307(23-O-[alpha-L-(4'-acetylrhamnopyranosyl]imberbic a...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295306(1-O-[alpha-L-(Rhamnopyranosyl]-23-acetoxyimberbic ...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295305(23-O-[alpha-L-(4'-Acetylrhamnopyranosyl]-3beta-ace...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295311(CHEMBL555367 | lantadene B)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295303(23-Acetoxyimberbic acid 29-methyl ester | CHEMBL55...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50295304(23-O-[alpha-L-(3',4'-Diacetylrhamnopyranosyl]-3bet...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to Bcl-xL by fluorescein-labeled Bak-BH3 peptide competition binding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed