Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50030470
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296598((R)-2-(2,4-dichlorophenylsulfonamido)-3-(thiophene...)
Affinity DataIC50:  8nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296610((R)-3-(1-methyl-1H-pyrazole-5-carboxamido)-2-(2,4,...)
Affinity DataIC50:  11nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296635((R)-2-(2,3-dichlorophenylsulfonamido)-3-(thiophene...)
Affinity DataIC50:  19nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296597((R)-3-(thiophene-3-carboxamido)-2-(2,4,6-trichloro...)
Affinity DataIC50:  24nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296603((R)-3-benzamido-2-(2-iodophenylsulfonamido)propano...)
Affinity DataIC50:  25nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296611((R)-3-(furan-3-carboxamido)-2-(2,4,6-trimethylphen...)
Affinity DataIC50:  32nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296609((R)-3-(2-methyloxazole-4-carboxamido)-2-(2,4,6-tri...)
Affinity DataIC50:  41nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296612((R)-3-(thiophene-3-carboxamido)-2-(2,4,6-trimethyl...)
Affinity DataIC50:  44nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296600((R)-3-benzamido-2-(2,3-dichlorophenylsulfonamido)p...)
Affinity DataIC50:  62nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296607((R)-3-(pyrimidine-5-carboxamido)-2-(2,4,6-trimethy...)
Affinity DataIC50:  63nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296632((R)-3-(2-methoxybenzamido)-2-(2,4,6-trimethylpheny...)
Affinity DataIC50:  78nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296608((R)-3-(nicotinamido)-2-(2,4,6-trimethylphenylsulfo...)
Affinity DataIC50:  81nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296596((R)-2-(3-cyanophenylsulfonamido)-3-(furan-3-carbox...)
Affinity DataIC50:  98nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296599((R)-3-benzamido-2-(2,6-dichlorophenylsulfonamido)p...)
Affinity DataIC50:  118nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296623((R)-3-benzamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50:  120nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296595((R)-3-(furan-3-carboxamido)-2-(3-methoxyphenylsulf...)
Affinity DataIC50:  208nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296633((R)-3-(furan-3-carboxamido)-2-(2-methylphenylsulfo...)
Affinity DataIC50:  260nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296604((R)-3-benzamido-2-(2-chlorophenylsulfonamido)propa...)
Affinity DataIC50:  260nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296606((R)-3-(isonicotinamido)-2-(2,4,6-trimethylphenylsu...)
Affinity DataIC50:  301nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296605((R)-3-benzamido-2-(2-methylphenylsulfonamido)propa...)
Affinity DataIC50:  320nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296634((R)-3-(furan-3-carboxamido)-2-(2-methoxyphenylsulf...)
Affinity DataIC50:  700nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296601((R)-3-benzamido-2-(2-methoxyphenylsulfonamido)prop...)
Affinity DataIC50:  729nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296594((R)-3-(furan-3-carboxamido)-2-(pyridine-3-sulfonam...)
Affinity DataIC50:  793nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296629((R)-3-acetamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50:  800nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296631((R)-3-(1-oxoisoindolin-2-yl)-2-(2,4,6-trimethylphe...)
Affinity DataIC50:  975nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296633((R)-3-(furan-3-carboxamido)-2-(2-methylphenylsulfo...)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of fibrinogen binding to alpha2beta3a integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296602((R)-3-benzamido-2-(2-(methylsulfonyl)phenylsulfona...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296630((R)-3-(2-(furan-3-yl)-2-oxoethylamino)-2-(2,4,6-tr...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296620((S)-3-acetamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296619((R)-3-acetamido-2-(phenylsulfonamido)propanoic aci...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296627((R)-3-butyramido-2-(2,4,6-trimethylphenylsulfonami...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296628((R)-3-amino-2-(2,4,6-trimethylphenylsulfonamido)pr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296626((R)-3-(tert-butoxycarbonylamino)-2-(2,4,6-trimethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296625((R)-3-(methoxycarbonylamino)-2-(2,4,6-trimethylphe...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296624((R)-3-(methylsulfonamido)-2-(2,4,6-trimethylphenyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296622((R)-3-(2-phenylacetamido)-2-(2,4,6-trimethylphenyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296621((R)-3-(benzylamino)-2-(2,4,6-trimethylphenylsulfon...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296618((R)-3-acetamido-2-(phenylmethylsulfonamido)propano...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296617((R)-3-acetamido-2-benzamidopropanoic acid | CHEMBL...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296616((R)-3-acetamido-2-(2,6-dichlorobenzamido)propanoic...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296614((R)-3-acetamido-2-(tert-butoxycarbonylamino)propan...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296613((R)-3-acetamido-2-(N,2,4,6-tetramethylphenylsulfon...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296615((R)-3-acetamido-2-(phenoxycarbonylamino)propanoic ...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50296634((R)-3-(furan-3-carboxamido)-2-(2-methoxyphenylsulf...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of fibrinogen binding to alpha2beta3a integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed