Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50030470
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296598BDBM50296598((R)-2-(2,4-dichlorophenylsulfonamido)-3-(thiophene...)
Affinity DataIC50: 8nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296610BDBM50296610((R)-3-(1-methyl-1H-pyrazole-5-carboxamido)-2-(2,4,...)
Affinity DataIC50: 11nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296635BDBM50296635((R)-2-(2,3-dichlorophenylsulfonamido)-3-(thiophene...)
Affinity DataIC50: 19nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296597BDBM50296597((R)-3-(thiophene-3-carboxamido)-2-(2,4,6-trichloro...)
Affinity DataIC50: 24nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296603BDBM50296603((R)-3-benzamido-2-(2-iodophenylsulfonamido)propano...)
Affinity DataIC50: 25nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296611BDBM50296611((R)-3-(furan-3-carboxamido)-2-(2,4,6-trimethylphen...)
Affinity DataIC50: 32nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296609BDBM50296609((R)-3-(2-methyloxazole-4-carboxamido)-2-(2,4,6-tri...)
Affinity DataIC50: 41nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296612BDBM50296612((R)-3-(thiophene-3-carboxamido)-2-(2,4,6-trimethyl...)
Affinity DataIC50: 44nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296600BDBM50296600((R)-3-benzamido-2-(2,3-dichlorophenylsulfonamido)p...)
Affinity DataIC50: 62nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296607BDBM50296607((R)-3-(pyrimidine-5-carboxamido)-2-(2,4,6-trimethy...)
Affinity DataIC50: 63nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296632BDBM50296632((R)-3-(2-methoxybenzamido)-2-(2,4,6-trimethylpheny...)
Affinity DataIC50: 78nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296608BDBM50296608((R)-3-(nicotinamido)-2-(2,4,6-trimethylphenylsulfo...)
Affinity DataIC50: 81nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296596BDBM50296596((R)-2-(3-cyanophenylsulfonamido)-3-(furan-3-carbox...)
Affinity DataIC50: 98nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296599BDBM50296599((R)-3-benzamido-2-(2,6-dichlorophenylsulfonamido)p...)
Affinity DataIC50: 118nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296623BDBM50296623((R)-3-benzamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50: 120nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296595BDBM50296595((R)-3-(furan-3-carboxamido)-2-(3-methoxyphenylsulf...)
Affinity DataIC50: 208nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296633BDBM50296633((R)-3-(furan-3-carboxamido)-2-(2-methylphenylsulfo...)
Affinity DataIC50: 260nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296604BDBM50296604((R)-3-benzamido-2-(2-chlorophenylsulfonamido)propa...)
Affinity DataIC50: 260nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296606BDBM50296606((R)-3-(isonicotinamido)-2-(2,4,6-trimethylphenylsu...)
Affinity DataIC50: 301nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296605BDBM50296605((R)-3-benzamido-2-(2-methylphenylsulfonamido)propa...)
Affinity DataIC50: 320nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296634BDBM50296634((R)-3-(furan-3-carboxamido)-2-(2-methoxyphenylsulf...)
Affinity DataIC50: 700nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296601BDBM50296601((R)-3-benzamido-2-(2-methoxyphenylsulfonamido)prop...)
Affinity DataIC50: 729nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296594BDBM50296594((R)-3-(furan-3-carboxamido)-2-(pyridine-3-sulfonam...)
Affinity DataIC50: 793nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296629BDBM50296629((R)-3-acetamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50: 800nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296631BDBM50296631((R)-3-(1-oxoisoindolin-2-yl)-2-(2,4,6-trimethylphe...)
Affinity DataIC50: 975nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-2(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296633BDBM50296633((R)-3-(furan-3-carboxamido)-2-(2-methylphenylsulfo...)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of fibrinogen binding to alpha2beta3a integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296602BDBM50296602((R)-3-benzamido-2-(2-(methylsulfonyl)phenylsulfona...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296630BDBM50296630((R)-3-(2-(furan-3-yl)-2-oxoethylamino)-2-(2,4,6-tr...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296620BDBM50296620((S)-3-acetamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296619BDBM50296619((R)-3-acetamido-2-(phenylsulfonamido)propanoic aci...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296627BDBM50296627((R)-3-butyramido-2-(2,4,6-trimethylphenylsulfonami...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296616BDBM50296616((R)-3-acetamido-2-(2,6-dichlorobenzamido)propanoic...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296617BDBM50296617((R)-3-acetamido-2-benzamidopropanoic acid | CHEMBL...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296614BDBM50296614((R)-3-acetamido-2-(tert-butoxycarbonylamino)propan...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296615BDBM50296615((R)-3-acetamido-2-(phenoxycarbonylamino)propanoic ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296621BDBM50296621((R)-3-(benzylamino)-2-(2,4,6-trimethylphenylsulfon...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296618BDBM50296618((R)-3-acetamido-2-(phenylmethylsulfonamido)propano...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296624BDBM50296624((R)-3-(methylsulfonamido)-2-(2,4,6-trimethylphenyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296625BDBM50296625((R)-3-(methoxycarbonylamino)-2-(2,4,6-trimethylphe...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296622BDBM50296622((R)-3-(2-phenylacetamido)-2-(2,4,6-trimethylphenyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296628BDBM50296628((R)-3-amino-2-(2,4,6-trimethylphenylsulfonamido)pr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296613BDBM50296613((R)-3-acetamido-2-(N,2,4,6-tetramethylphenylsulfon...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-V(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296626BDBM50296626((R)-3-(tert-butoxycarbonylamino)-2-(2,4,6-trimethy...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetIntegrin alpha-2(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50296634BDBM50296634((R)-3-(furan-3-carboxamido)-2-(2-methoxyphenylsulf...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of fibrinogen binding to alpha2beta3a integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed