Compile Data Set for Download or QSAR
maximum 50k data
Found 142 Enz. Inhib. hit(s) with all data for entry = 50030475
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296761(CHEMBL564105 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296768(CHEMBL554908 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296755(CHEMBL558452 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296773(6-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296767(CHEMBL563901 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296772(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296769(CHEMBL552069 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296754(CHEMBL558647 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296779(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296781(6-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296762(CHEMBL550114 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296765(CHEMBL558322 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296774((R)-3-amino-1-((S)-2-((4-(trifluoromethyl)pyrimidi...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296780(6-((((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)b...)
Affinity DataIC50:  4nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296766(CHEMBL557723 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296776((R)-3-amino-1-((S)-2-((pyrimidin-2-ylamino)methyl)...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296756(CHEMBL559602 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296763(CHEMBL557860 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296771((R)-3-amino-1-((S)-2-((2-(trifluoromethyl)pyrimidi...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296778((R)-3-amino-1-((S)-2-((5-fluoropyridin-2-ylamino)m...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296764(CHEMBL558323 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296760(CHEMBL550321 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296775((R)-3-amino-1-((S)-2-((5-fluoropyrimidin-2-ylamino...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296759(CHEMBL559601 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296120(CHEMBL563272 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  8nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296133(CHEMBL563648 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  9nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296770((R)-3-amino-1-((S)-2-((cyclopropylmethoxy)methyl)p...)
Affinity DataIC50:  10nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296757(CHEMBL564283 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  12nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296777((R)-3-amino-1-((S)-2-((6-(trifluoromethyl)pyridin-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296758(CHEMBL559543 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  27nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296754(CHEMBL558647 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296775((R)-3-amino-1-((S)-2-((5-fluoropyrimidin-2-ylamino...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296759(CHEMBL559601 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296781(6-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  340nMAssay Description:Inhibition of DPP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296777((R)-3-amino-1-((S)-2-((6-(trifluoromethyl)pyridin-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human recombinant DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296774((R)-3-amino-1-((S)-2-((4-(trifluoromethyl)pyrimidi...)
Affinity DataIC50:  400nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296756(CHEMBL559602 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  470nMAssay Description:Inhibition of human recombinant DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296777((R)-3-amino-1-((S)-2-((6-(trifluoromethyl)pyridin-...)
Affinity DataIC50:  530nMAssay Description:Inhibition of DPP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296780(6-((((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)b...)
Affinity DataIC50:  600nMAssay Description:Inhibition of DPP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296779(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  700nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296779(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  700nMAssay Description:Inhibition of DPP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296778((R)-3-amino-1-((S)-2-((5-fluoropyridin-2-ylamino)m...)
Affinity DataIC50:  800nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296755(CHEMBL558452 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  880nMAssay Description:Inhibition of human recombinant DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296778((R)-3-amino-1-((S)-2-((5-fluoropyridin-2-ylamino)m...)
Affinity DataIC50:  890nMAssay Description:Inhibition of DPP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296780(6-((((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)b...)
Affinity DataIC50:  900nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296780(6-((((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)b...)
Affinity DataIC50:  990nMAssay Description:Inhibition of human recombinant DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296772(2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)bu...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296757(CHEMBL564283 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant DPP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296761(CHEMBL564105 | N-(((S)-1-((R)-3-amino-4-(2,4,5-tri...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of CYP2D6 in human human liver microsomes by mass spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Santhera Pharmaceuticals (Switzerland)

Curated by ChEMBL
LigandPNGBDBM50296777((R)-3-amino-1-((S)-2-((6-(trifluoromethyl)pyridin-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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