Compile Data Set for Download or QSAR
maximum 50k data
Found 129 Enz. Inhib. hit(s) with all data for entry = 50030599
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298862(4-((S)-3-(methylamino)-2-((R)-2-((4-methylcyclohex...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298864(4-((2S)-2-((2R)-2-(2-(bicyclo[2.2.1]heptan-2-yl)et...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298857(4-((S)-2-(cycloheptylmethylamino)-3-((S)-1-(4-hydr...)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298865(4-((S)-2-((R)-2-(cycloheptylmethylamino)pentylamin...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298863(4-{(S)-2-[(R)-2-(2-Adamantan-1-yl-ethylamino)-pent...)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298857(4-((S)-2-(cycloheptylmethylamino)-3-((S)-1-(4-hydr...)
Affinity DataIC50:  54nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298895((2S,3S)-2-((R)-4-(3-cyclohexylpropyl)-3-isopropylp...)
Affinity DataIC50:  58nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298889((R)-4-(2-(4-(cycloheptylmethyl)piperazin-1-yl)-3-(...)
Affinity DataIC50:  89nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298890(4-((2R)-2-(4-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)p...)
Affinity DataIC50:  91nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298884((S)-4-(2-(4-(cycloheptylmethyl)piperazin-1-yl)-3-(...)
Affinity DataIC50:  93nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298861(4-((S)-2-((R)-2-(2-cyclopentylethylamino)pentylami...)
Affinity DataIC50:  98nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298858(4-((S)-2-((S)-3-(4-hydroxyphenyl)-2-((4-methylcycl...)
Affinity DataIC50:  102nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298874((R)-N2-(2-cyclopentylethyl)-N1-((R)-1-(methylamino...)
Affinity DataIC50:  102nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298882(4-(((R)-4-((R)-1-(benzylamino)hexan-2-yl)-1-isobut...)
Affinity DataIC50:  102nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298866(4-((S)-2-(cycloheptylmethylamino)-3-((R)-1-(methyl...)
Affinity DataIC50:  107nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298896(CHEMBL573347 | {(S)-2-[(R)-4-(2-Adamantan-1-yl-eth...)
Affinity DataIC50:  119nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298884((S)-4-(2-(4-(cycloheptylmethyl)piperazin-1-yl)-3-(...)
Affinity DataIC50:  152nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298883(4-(((R)-4-((R)-1-(benzylamino)hexan-2-yl)-1-(cyclo...)
Affinity DataIC50:  161nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298885(4-((2S)-2-(4-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)p...)
Affinity DataIC50:  167nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298860(4-((S)-2-(2-cyclopentylethylamino)-3-((S)-1-(4-hyd...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298864(4-((2S)-2-((2R)-2-(2-(bicyclo[2.2.1]heptan-2-yl)et...)
Affinity DataIC50:  174nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298868(4-((2S)-2-(2-(bicyclo[2.2.1]heptan-2-yl)ethylamino...)
Affinity DataIC50:  178nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298860(4-((S)-2-(2-cyclopentylethylamino)-3-((S)-1-(4-hyd...)
Affinity DataIC50:  186nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298886(4-((S)-2-((S)-3-isopropyl-4-(3-methylphenethyl)pip...)
Affinity DataIC50:  206nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298889((R)-4-(2-(4-(cycloheptylmethyl)piperazin-1-yl)-3-(...)
Affinity DataIC50:  223nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298887(4-((2S)-2-((3S)-4-(2-(bicyclo[2.2.1]heptan-2-yl)et...)
Affinity DataIC50:  223nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298867(4-((S)-3-((R)-1-(methylamino)pentan-2-ylamino)-2-(...)
Affinity DataIC50:  225nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298856(4-((2R)-2-((3R)-4-(2-(bicyclo[2.2.1]heptan-2-yl)et...)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298865(4-((S)-2-((R)-2-(cycloheptylmethylamino)pentylamin...)
Affinity DataIC50:  238nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298869(4-((S)-2-(2-cyclopentylethylamino)-3-((R)-1-(methy...)
Affinity DataIC50:  240nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298859(4-((2S)-2-(2-(bicyclo[2.2.1]heptan-2-yl)ethylamino...)
Affinity DataIC50:  270nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298858(4-((S)-2-((S)-3-(4-hydroxyphenyl)-2-((4-methylcycl...)
Affinity DataIC50:  313nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298868(4-((2S)-2-(2-(bicyclo[2.2.1]heptan-2-yl)ethylamino...)
Affinity DataIC50:  333nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298856(4-((2R)-2-((3R)-4-(2-(bicyclo[2.2.1]heptan-2-yl)et...)
Affinity DataIC50:  336nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298885(4-((2S)-2-(4-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)p...)
Affinity DataIC50:  373nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298887(4-((2S)-2-((3S)-4-(2-(bicyclo[2.2.1]heptan-2-yl)et...)
Affinity DataIC50:  374nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298881(4-((R)-3-(benzylamino)-2-((S)-4-(3,3-dimethylbutyl...)
Affinity DataIC50:  387nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298866(4-((S)-2-(cycloheptylmethylamino)-3-((R)-1-(methyl...)
Affinity DataIC50:  439nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298859(4-((2S)-2-(2-(bicyclo[2.2.1]heptan-2-yl)ethylamino...)
Affinity DataIC50:  457nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298888((R)-4-(3-(methylamino)-2-(4-(4-methylpentyl)pipera...)
Affinity DataIC50:  471nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298890(4-((2R)-2-(4-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)p...)
Affinity DataIC50:  476nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298863(4-{(S)-2-[(R)-2-(2-Adamantan-1-yl-ethylamino)-pent...)
Affinity DataIC50:  530nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298861(4-((S)-2-((R)-2-(2-cyclopentylethylamino)pentylami...)
Affinity DataIC50:  648nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298855(4-((R)-2-((R)-4-(3-cyclohexylpropyl)-3-isopropylpi...)
Affinity DataIC50:  654nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298869(4-((S)-2-(2-cyclopentylethylamino)-3-((R)-1-(methy...)
Affinity DataIC50:  766nMAssay Description:Displacement of [3H]U69593 from guinea pig kappa opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298855(4-((R)-2-((R)-4-(3-cyclohexylpropyl)-3-isopropylpi...)
Affinity DataIC50:  920nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298871((R)-N1-methyl-N2-((R)-2-((4-methylcyclohexyl)methy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298872((R)-N*2*-(2-Adamantan-1-yl-ethyl)-N*1*-((R)-1-meth...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298873((2R)-N2-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)-N1-((...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50298874((R)-N2-(2-cyclopentylethyl)-N1-((R)-1-(methylamino...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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