Compile Data Set for Download or QSAR
Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50030705
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132713BDBM50132713(Methyl arachidonoyl fluorophophonate | methyl -ico...)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60622BDBM60622(BDBM50300355 | US9133148, A | US11753371, Compound...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059523BDBM50059523(Arachidonyltrifluoromethane | (6Z,9Z,12Z,15Z)-1,1,...)
Affinity DataIC50: 12.3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132713BDBM50132713(Methyl arachidonoyl fluorophophonate | methyl -ico...)
Affinity DataIC50: 26.3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26736BDBM26736(N,N-dimethyl-5-[(4-phenylphenyl)methyl]-1H-1,2,3,4...)
Affinity DataIC50: 37.3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26736BDBM26736(N,N-dimethyl-5-[(4-phenylphenyl)methyl]-1H-1,2,3,4...)
Affinity DataIC50: 54.4nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300344BDBM50300344(1-Biphenyl-4-ylmethylmaleimide | CHEMBL576859)
Affinity DataIC50: 790nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300346BDBM50300346(N-Oleylmaleimide | CHEMBL566336)
Affinity DataIC50: 930nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60419BDBM60419(NAM | BDBM50295658)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300339BDBM50300339(1-Biphenyl-2-ylmaleimide | CHEMBL567440)
Affinity DataIC50: 1.55E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300341BDBM50300341(1-Biphenyl-4-ylmaleimide | CHEMBL567545)
Affinity DataIC50: 1.62E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300349BDBM50300349(1,4-bis(malimido)xylene | CHEMBL565711)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300351BDBM50300351(cid_20992 | CHEMBL567422 | (1-(6-(2,5-dioxo-2H-pyr...)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300352BDBM50300352(1,8-bis-maleimidodiethyleneglycol | CHEMBL575383)
Affinity DataIC50: 1.95E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300316BDBM50300316(1-(2-Ethylphenyl)maleimide | CHEMBL574140)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300347BDBM50300347(phenyl-1,3-bismaleimide | CHEMBL573689)
Affinity DataIC50: 2.03E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300322BDBM50300322(1-(4-Heptylphenyl)maleimide | CHEMBL565892)
Affinity DataIC50: 2.12E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300342BDBM50300342(1-(4-phenylbutyl)-1H-pyrrole-2,5-dione | 1-(4-Phen...)
Affinity DataIC50: 2.14E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60419BDBM60419(NAM | BDBM50295658)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300348BDBM50300348(phenyl-1,4-bismaleimide | CHEMBL576594)
Affinity DataIC50: 2.22E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270000BDBM50270000(1,1-(Methylene-di-1,4-phenylene)-bismaleimide | 1,...)
Affinity DataIC50: 2.24E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300337BDBM50300337(1-(3-Iodophenyl)maleimide | CHEMBL565710)
Affinity DataIC50: 2.24E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300340BDBM50300340(cid_930984 | CHEMBL567622 | 1-Biphenyl-3-ylmaleimi...)
Affinity DataIC50: 2.34E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300328BDBM50300328(1-(3-Fluorophenyl)maleimide | CHEMBL574358)
Affinity DataIC50: 2.39E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300313BDBM50300313(1-(2-Methylphenyl)maleimide | CHEMBL578794)
Affinity DataIC50: 2.69E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300345BDBM50300345(N-Palmitylmaleimide | CHEMBL568289)
Affinity DataIC50: 2.69E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300314BDBM50300314(1-(3-Methylphenyl)maleimide | CHEMBL567421)
Affinity DataIC50: 2.75E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300331BDBM50300331(1-(3-Chlorophenyl)maleimide | CHEMBL578977)
Affinity DataIC50: 2.82E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300318BDBM50300318(1-(4-Ethylphenyl)maleimide | CHEMBL577071)
Affinity DataIC50: 2.82E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300321BDBM50300321(1-(4-Isopropylphenyl)maleimide | CHEMBL576625)
Affinity DataIC50: 2.88E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300333BDBM50300333(1-(2-Bromophenyl)maleimide | CHEMBL578978)
Affinity DataIC50: 2.92E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300343BDBM50300343(1-(4-Ethylbenzyl)maleimide | CHEMBL576626)
Affinity DataIC50: 3.55E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50050711BDBM50050711(1-Nonyl-pyrrole-2,5-dione | N-Nonylmaleimide | CHE...)
Affinity DataIC50: 3.55E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60622BDBM60622(BDBM50300355 | US9133148, A | US11753371, Compound...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300330BDBM50300330(1-(2-Chlorophenyl)maleimide | CHEMBL565700)
Affinity DataIC50: 4.17E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300334BDBM50300334(1-(3-Bromophenyl)maleimide | CHEMBL583957)
Affinity DataIC50: 4.27E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300338BDBM50300338(1-(4-Iodophenyl)maleimide | CHEMBL579183)
Affinity DataIC50: 4.34E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300335BDBM50300335(1-(4-Bromophenyl)maleimide | CHEMBL566998)
Affinity DataIC50: 4.37E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300327BDBM50300327(1-(2-Fluorophenyl)maleimide | CHEMBL579012)
Affinity DataIC50: 4.47E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300317BDBM50300317(1-(3-Ethylphenyl)maleimide | CHEMBL568527)
Affinity DataIC50: 4.68E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300336BDBM50300336(1-(2-Iodophenyl)maleimide | CHEMBL566999)
Affinity DataIC50: 5.01E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7804BDBM7804(1-benzyl-2,5-dihydro-1H-pyrrole-2,5-dione | Maleim...)
Affinity DataIC50: 5.14E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300329BDBM50300329(1-(4-Fluorophenyl)maleimide | CHEMBL583956)
Affinity DataIC50: 5.18E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128581BDBM50128581(cyclohexyl biphenyl-3-ylcarbamate | CHEMBL77767 | ...)
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300326BDBM50300326(1-(4-Methoxyphenyl)maleimide | CHEMBL568288)
Affinity DataIC50: 5.75E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300341BDBM50300341(1-Biphenyl-4-ylmaleimide | CHEMBL567545)
Affinity DataIC50: 5.89E+3nMAssay Description:Displacement of [3H]ethanolamine from human recombinant FAAH by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300319BDBM50300319(1-(4-Propylphenyl)maleimide | CHEMBL568528)
Affinity DataIC50: 5.89E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059523BDBM50059523(Arachidonyltrifluoromethane | (6Z,9Z,12Z,15Z)-1,1,...)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300325BDBM50300325(1-(3-Methoxyphenyl)maleimide | CHEMBL566111)
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Louvain Drug Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300324BDBM50300324(1-(2-Methoxyphenyl)maleimide | CHEMBL565904)
Affinity DataIC50: 6.92E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
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