Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50030753
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 5nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300888((S)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)
Affinity DataIC50: 6nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300885(N-sec-butyl-4-(3-(4-fluorophenyl)-5-isopropylisoxa...)
Affinity DataIC50: 30nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 40nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)
Affinity DataIC50: 47nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM13531(4-[4-(4-Fluorophenyl)-5-(4-pyridinyl)-1H-imidazol-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300886(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)-N-...)
Affinity DataIC50: 60nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)
Affinity DataIC50: 90nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 120nMAssay Description:Inhibition of CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50: 230nMAssay Description:Inhibition of CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50: 230nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300889(N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)...)
Affinity DataIC50: 300nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50229971(4-[4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-5-pyridin...)
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-fused rat CK1delta expressed in Escherichia coli using phosphorylated peptide TFRPRTSpSNASTIS as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300889(N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)...)
Affinity DataIC50: 330nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300891((rac)-N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol...)
Affinity DataIC50: 340nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50: 447nMAssay Description:Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300887((R)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)
Affinity DataIC50: 450nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50: 450nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50: 540nMAssay Description:Inhibition of JNK3 by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300889(N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)...)
Affinity DataIC50: 700nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300891((rac)-N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol...)
Affinity DataIC50: 820nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300891((rac)-N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol...)
Affinity DataIC50: 890nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50263829(3-[(2,4,6-trimethoxyphenyl)methylidenyl]-indolin-2...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human CK1deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of JNK2 by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300888((S)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206423(4-(5-(4-fluorophenyl)-3-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300886(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)-N-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)
Affinity DataIC50: 2.52E+3nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50229971(4-[4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-5-pyridin...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of GST-fused human p38alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed