Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50038874
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 5nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294138(N-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13R,14R,16S,17S)-...)
Affinity DataIC50: 5.70nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294160(N-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-11,...)
Affinity DataIC50: 8.30nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294146(N-(5-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-...)
Affinity DataIC50: 8.5nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294153(3-acetamido-N-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-...)
Affinity DataIC50: 9.30nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294159(N-(2-(3-(2-(2-((8S,9R,10S,11S,13S,14S,16R,17R)-9-f...)
Affinity DataIC50: 9.80nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294147(N-(5-(5-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluo...)
Affinity DataIC50: 12nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294137(CHEMBL556523)
Affinity DataIC50: 14nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294139(N-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13R,14R,16S,17...)
Affinity DataIC50: 14nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294157(1-(2-(2-((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-...)
Affinity DataIC50: 15nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294149(N-(5-(5-(5-(5-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-...)
Affinity DataIC50: 16nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294150(N-(4-(5-(5-(5-(5-(1-((8S,9R,10S,11S,13S,14S,16R,17...)
Affinity DataIC50: 16nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294148(N-(5-(5-(5-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-9-f...)
Affinity DataIC50: 20nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294152(CHEMBL563739)
Affinity DataIC50: 20nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294143(N-(5-(4-(5-(5-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13...)
Affinity DataIC50: 21nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294144(N-(5-(5-(4-(5-(5-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R...)
Affinity DataIC50: 21nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294151(N-(5-(4-(5-(5-(5-(5-(1-((8S,9R,10S,11S,13S,14S,16R...)
Affinity DataIC50: 22nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294142(N-(4-(5-(5-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13R,1...)
Affinity DataIC50: 23nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294140(N-(5-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13R,14R,16S...)
Affinity DataIC50: 26nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294145(CHEMBL564923)
Affinity DataIC50: 27nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294141(N-(5-(5-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13R,14R,...)
Affinity DataIC50: 34nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294158(N-(5-(2-((8R,9S,10R,11R,13R,14R,16S,17S)-9-fluoro-...)
Affinity DataIC50: 460nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294154(N-(5-(5-(2-((8R,9S,10R,11R,13R,14R,16S,17S)-9-fluo...)
Affinity DataIC50: 480nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294155(N-(5-(5-(5-(2-((8R,9S,10R,11R,13R,14R,16S,17S)-9-f...)
Affinity DataIC50: 550nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50271344((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-11,17-dih...)
Affinity DataIC50: 600nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294156(N-(5-(5-(5-(4-(5-(5-(5-(5-(2-((8R,9S,10R,11R,13R,1...)
Affinity DataIC50: 840nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed