Compile Data Set for Download or QSAR
maximum 50k data
Found 53 Enz. Inhib. hit(s) with all data for entry = 50030494
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297070(CHEMBL560474 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297062(4-(5-chloropyridin-2-yl)-N-(2-cyclopropyl-3-methyl...)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297073(CHEMBL564106 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297061(CHEMBL551934 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297059(CHEMBL561134 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297067(CHEMBL565105 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297071(CHEMBL562136 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297068(CHEMBL551470 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  4.40nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297042(CHEMBL557731 | N-(2-methylimidazo[1,2-a]pyridin-6-...)
Affinity DataIC50:  4.60nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297052(CHEMBL563725 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  4.80nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297064(CHEMBL563728 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  4.80nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297041(CHEMBL557664 | N-(2-isopropylimidazo[1,2-a]pyridin...)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297063(CHEMBL559680 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297044(CHEMBL557730 | N-(2-cyclopropylimidazo[1,2-a]pyrid...)
Affinity DataIC50:  5.60nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297065(CHEMBL563096 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297072(CHEMBL558826 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  6.80nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297045(CHEMBL549512 | N-(2-tert-butylimidazo[1,2-a]pyridi...)
Affinity DataIC50:  7.10nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297058(CHEMBL556432 | N-(2-cyclopropylimidazo[1,2-a]pyrid...)
Affinity DataIC50:  8.20nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297055(CHEMBL562074 | N-(2-cyclopropyl-3-(hydroxymethyl)i...)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297043(CHEMBL554287 | N-(2-propylimidazo[1,2-a]pyridin-6-...)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297049(CHEMBL560334 | N-(2-(2-hydroxypropan-2-yl)imidazo[...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297068(CHEMBL551470 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297061(CHEMBL551934 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297053(CHEMBL551332 | N-(2-cyclopropyl-3-ethylimidazo[1,2...)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297072(CHEMBL558826 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297048(CHEMBL556296 | N-(2-(1-hydroxyethyl)imidazo[1,2-a]...)
Affinity DataIC50:  30nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297051(CHEMBL551408 | N-(2-((N-methylacetamido)methyl)imi...)
Affinity DataIC50:  35nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297076(CHEMBL559801 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  44nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297066(CHEMBL563836 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  48nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297070(CHEMBL560474 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  59nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297075(CHEMBL558326 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  61nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297073(CHEMBL564106 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297050(CHEMBL563984 | N-(2-((dimethylamino)methyl)imidazo...)
Affinity DataIC50:  83nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297064(CHEMBL563728 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  85nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297063(CHEMBL559680 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297066(CHEMBL563836 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  94nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297071(CHEMBL562136 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  94nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297062(4-(5-chloropyridin-2-yl)-N-(2-cyclopropyl-3-methyl...)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297074(CHEMBL563156 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  102nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297067(CHEMBL565105 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  109nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297076(CHEMBL559801 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  121nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297065(CHEMBL563096 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  122nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297047(CHEMBL563147 | N-(2-(hydroxymethyl)imidazo[1,2-a]p...)
Affinity DataIC50:  130nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297060(CHEMBL557317 | N-(2-cyclopropylimidazo[1,2-a]pyrid...)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297069(CHEMBL549583 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  160nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297074(CHEMBL563156 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  164nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297075(CHEMBL558326 | N-(2-cyclopropyl-3-methylimidazo[1,...)
Affinity DataIC50:  217nMAssay Description:Antagonist activity at human MCH1 receptor expressed in CHO cells assessed as inhibition of MCH-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297054(CHEMBL562073 | N-(2,3-dicyclopropylimidazo[1,2-a]p...)
Affinity DataIC50:  260nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297040(CHEMBL560677 | N-(imidazo[1,2-a]pyridin-6-yl)-4'-(...)
Affinity DataIC50:  300nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297056(CHEMBL561133 | N-(3-acetyl-2-cyclopropylimidazo[1,...)
Affinity DataIC50:  320nMAssay Description:Displacement of [125I]MCH from human MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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