Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50030790
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  33nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301422(CHEMBL572030 | vinyl 3-(4-(3-chlorophenylamino)qui...)
Affinity DataIC50:  180nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301421((3-(4-(3-chlorophenylamino)quinazolin-6-yl)-1-meth...)
Affinity DataIC50:  240nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301426(CHEMBL583683 | chloromethyl 3-(4-(3-chlorophenylam...)
Affinity DataIC50:  390nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301424(2-chloroethyl 3-(4-(3-chlorophenylamino)quinazolin...)
Affinity DataIC50:  500nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301425(CHEMBL572028 | acetoxymethyl 3-(4-(3-chlorophenyla...)
Affinity DataIC50:  630nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301423(CHEMBL572031 | vinyl 3-(4-(3-chlorophenylamino)qui...)
Affinity DataIC50:  720nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301427(4-nitrophenyl 3-(4-(3-chlorophenylamino)quinazolin...)
Affinity DataIC50:  770nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed