Compile Data Set for Download or QSAR
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Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50030802
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301693(5-(5-((4-(dimethylamino)piperidin-1-yl)methyl)fura...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301694(5-(5-((4-isopropylpiperazin-1-yl)methyl)furan-3-yl...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301679(4-(4-methyl-1H-indol-5-ylamino)-5-(3-((4-methylpip...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301695(5-(5-((4-cyclopentylpiperazin-1-yl)methyl)furan-3-...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301685(1-((4-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301678(4-(4-methyl-1H-indol-5-ylamino)-5-(4-((4-methylpip...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301684(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301676(5-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301689(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(thiomorpholi...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301688(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(morpholinome...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301693(5-(5-((4-(dimethylamino)piperidin-1-yl)methyl)fura...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301675(5-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301680(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(morpholinome...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301685(1-((4-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  9.70nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301687(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C epsilon type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PKCepsilon by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301694(5-(5-((4-isopropylpiperazin-1-yl)methyl)furan-3-yl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301695(5-(5-((4-cyclopentylpiperazin-1-yl)methyl)furan-3-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301679(4-(4-methyl-1H-indol-5-ylamino)-5-(3-((4-methylpip...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301681(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(morpholinome...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301678(4-(4-methyl-1H-indol-5-ylamino)-5-(4-((4-methylpip...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301676(5-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301691(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(pyrrolidin-1...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301687(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301682(4-(4-methyl-1H-indol-5-ylamino)-6'-((4-methylpiper...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301690(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(piperidin-1-...)
Affinity DataIC50:  41nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301692(5-(5-((diethylamino)methyl)furan-2-yl)-4-(4-methyl...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301684(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301675(5-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301680(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(morpholinome...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301681(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(morpholinome...)
Affinity DataIC50:  84nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301688(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(morpholinome...)
Affinity DataIC50:  86nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301689(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(thiomorpholi...)
Affinity DataIC50:  94nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C eta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  140nMAssay Description:Inhibition of PKCeta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301692(5-(5-((diethylamino)methyl)furan-2-yl)-4-(4-methyl...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301683(4-(4-methyl-1H-indol-5-ylamino)-5'-((4-methylpiper...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301677(5-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301682(4-(4-methyl-1H-indol-5-ylamino)-6'-((4-methylpiper...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301691(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(pyrrolidin-1...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301690(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(piperidin-1-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase Lck(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301677(5-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of PKCbeta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMAP kinase-activated protein kinase 2(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRho-associated protein kinase 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of ROCK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C zeta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PKCzeta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed