Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 5679
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  22nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92582(ETP-45798, 9)
Affinity DataIC50:  114nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM50328064(CHEMBL1258354 | ETP-7382 | N-(3-methoxyphenyl)-1-m...)
Affinity DataIC50:  400nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92586(ETP-45867, 14)
Affinity DataIC50:  840nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92584(ETP-45874, 11)
Affinity DataIC50:  970nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92583(ETP-45799, 10)
Affinity DataIC50:  1.66E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92588(ETP-45875, 16)
Affinity DataIC50:  3.53E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92574(ETP-5935)
Affinity DataIC50:  4.90E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92579(ETP-45419, 3d)
Affinity DataIC50:  5.51E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92587(ETP-45871, 15)
Affinity DataIC50:  5.80E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92589(ETP-45876, 17)
Affinity DataIC50:  7.00E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM50298309(CHEMBL574533 | ETP-7146 | N-(3-methoxyphenyl)-1-me...)
Affinity DataIC50:  9.20E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92575(ETP-6531)
Affinity DataIC50:  1.26E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92573(ETP-8162)
Affinity DataIC50:  1.26E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  1.31E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92581(ETP-45797, 7)
Affinity DataIC50:  1.61E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  1.68E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92576(ETP-45415, 3a)
Affinity DataIC50:  3.51E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92577(ETP-45416, 3b)
Affinity DataIC50:  3.68E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  3.98E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92580(ETP-45700, 6)
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92578(ETP-45654, 3c)
Affinity DataIC50: >5.00E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  1.29E+5nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  1.52E+5nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50:  7.17E+5nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed