Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50030732
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300648BDBM50300648(4-(3-((S)-1-((cis)-2-((S)-5-amino-1-(benzylamino)-...)
Affinity DataIC50: 68nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300658BDBM50300658(4-((E)-3-((S)-1-((1R,2S,5S)-2-(2-(benzyloxy)ethylc...)
Affinity DataIC50: 69nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300657BDBM50300657(4-(3-((S)-1-((cis)-2-((2R,3S)-6-amino-2-(benzyloxy...)
Affinity DataIC50: 69nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300656BDBM50300656(4-(3-((S)-1-((cis)-2-((S)-5-amino-1-(benzyloxy)-5-...)
Affinity DataIC50: 94nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300627BDBM50300627(4-(3-((S)-1-((S)-2-((R)-5-amino-5-oxopentan-2-ylca...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300646BDBM50300646(4-(3-((S)-4-methyl-1-oxo-1-((S)-2-(2-ureidoethylca...)
Affinity DataIC50: 131nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50198780BDBM50198780(pCinn-Leu-Pro-Gln-NHBn | 4-(3-((S)-1-((S)-2-((S)-5...)
Affinity DataIC50: 138nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300650BDBM50300650(4-(3-((S)-1-((cis)-2-((R)-5-amino-5-oxopentan-2-yl...)
Affinity DataIC50: 175nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300634BDBM50300634(4-(3-((S)-1-((S)-2-((2R,3S)-6-amino-2-(benzyloxy)-...)
Affinity DataIC50: 272nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50423685BDBM50423685(CHEMBL502473)
Affinity DataIC50: 290nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300655BDBM50300655((S)-5-amino-2-((cis)-3-((S)-4-methyl-2-(3-(4-(phos...)
Affinity DataIC50: 290nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300633BDBM50300633(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(benzyloxy)-5-ox...)
Affinity DataIC50: 294nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300649BDBM50300649(4-(3-((S)-1-((cis)-2-(4-amino-4-oxobutylcarbamoyl)...)
Affinity DataIC50: 303nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300642BDBM50300642(2-((S)-1-((S)-4-methyl-2-(3-(4-(phosphonooxy)pheny...)
Affinity DataIC50: 360nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50198778BDBM50198778(pCin-Leu-Pro-Ser(CONH2)-NHBn | (S)-3-(benzylamino)...)
Affinity DataIC50: 379nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300654BDBM50300654(4-(3-((S)-1-((cis)-2-((2R,3S)-6-amino-2-hydroxy-6-...)
Affinity DataIC50: 437nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300644BDBM50300644((R)-3-(benzyloxy)-2-((S)-1-((S)-4-methyl-2-(3-(4-(...)
Affinity DataIC50: 454nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300653BDBM50300653(4-(3-((S)-1-((cis)-2-((R)-1-amino-1-oxooctan-4-ylc...)
Affinity DataIC50: 499nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300651BDBM50300651(4-(3-((S)-1-((cis)-2-((S)-6-amino-2-methyl-6-oxohe...)
Affinity DataIC50: 511nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300618BDBM50300618(4-(3-((S)-1-((S)-2-(4-amino-4-oxobutylcarbamoyl)py...)
Affinity DataIC50: 574nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300641BDBM50300641(4-(3-((S)-1-((S)-2-((S)-1-acetamido-5-amino-5-oxop...)
Affinity DataIC50: 589nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300635BDBM50300635((S)-5-amino-2-((S)-1-((S)-4-methyl-2-(3-(4-(phosph...)
Affinity DataIC50: 615nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300643BDBM50300643((R)-2-((S)-1-((S)-4-methyl-2-(3-(4-(phosphonooxy)p...)
Affinity DataIC50: 797nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300632BDBM50300632(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(4-hydroxyphenyl...)
Affinity DataIC50: 848nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50198779BDBM50198779((2R,3S)-4-(benzylamino)-3-((S)-1-((S)-4-methyl-2-(...)
Affinity DataIC50: 850nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300614BDBM50300614(4-(3-((S)-1-((S)-2-((S)-4-amino-1-(benzylamino)-1,...)
Affinity DataIC50: 874nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300639BDBM50300639(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(dibenzylamino)-...)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300619BDBM50300619(4-(3-((S)-1-((S)-2-((E)-4-amino-4-oxobut-2-enylcar...)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300620BDBM50300620(4-(3-((S)-1-((S)-2-(4-amino-4-oxobut-2-ynylcarbamo...)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300628BDBM50300628(4-(3-((S)-1-((S)-2-((S)-5-amino-5-oxopentan-2-ylca...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300636BDBM50300636(4-(3-((S)-1-((S)-2-((S)-5-amino-5-oxo-1-(piperidin...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300640BDBM50300640((S)-5-amino-2-((S)-1-((S)-4-methyl-2-(3-(4-(phosph...)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300637BDBM50300637(4-(3-((S)-1-((S)-2-((S)-5-amino-1-(4-methylpiperaz...)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300631BDBM50300631(4-(3-((S)-1-((S)-2-((R)-1-amino-1-oxooctan-4-ylcar...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300647BDBM50300647(4-(3-((S)-4-methyl-1-oxo-1-((S)-2-((R)-1-ureidopro...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300615BDBM50300615(4-(3-((S)-1-((S)-2-((S)-6-amino-1-(benzylamino)-1,...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300638BDBM50300638(4-(3-((S)-1-((S)-2-((S)-5-amino-1-morpholino-5-oxo...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300652BDBM50300652(4-(3-((S)-1-((cis)-2-((S)-1-amino-6-methyl-1-oxohe...)
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300626BDBM50300626(4-(3-((S)-1-((S)-2-(4-hydrazinyl-4-oxobutylcarbamo...)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300629BDBM50300629(4-(3-((S)-1-((S)-2-((S)-6-amino-2-methyl-6-oxohexa...)
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300625BDBM50300625(4-(3-((S)-1-((S)-2-(4-(hydroxyamino)-4-oxobutylcar...)
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300622BDBM50300622(4-(3-((S)-1-((S)-2-((3S,5S)-5-carbamoylpyrrolidin-...)
Affinity DataIC50: 3.21E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300621BDBM50300621(4-(3-((S)-1-((S)-2-((S)-2-(3-amino-3-oxopropyl)pyr...)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300623BDBM50300623(4-(3-((S)-1-((S)-2-((3R,5S)-5-carbamoylpyrrolidin-...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300630BDBM50300630(4-(3-((S)-1-((S)-2-((S)-1-amino-6-methyl-1-oxohept...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300613BDBM50300613(4-(3-((S)-1-((S)-2-(2-(benzylamino)-2-oxoethylcarb...)
Affinity DataIC50: 4.94E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300645BDBM50300645((2S,3R)-3-(benzyloxy)-2-((S)-1-((S)-4-methyl-2-(3-...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300617BDBM50300617(4-(3-((S)-1-((S)-2-((S)-1-amino-1-oxopropan-2-ylca...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300616BDBM50300616(4-(3-((S)-1-((S)-2-carbamoylpyrrolidin-1-yl)-4-met...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSignal transducer and activator of transcription 3(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50300624BDBM50300624(4-(3-((S)-4-methyl-1-oxo-1-((S)-2-(3-sulfamoylprop...)
Affinity DataIC50: 6.82E+4nMAssay Description:Inhibition of Stat3 SH2 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed