Compile Data Set for Download or QSAR
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Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50039089
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310966(4-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  22nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310971(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(4-(2...)
Affinity DataIC50:  25nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310985(CHEMBL1078666 | N-(4-((3-bromo-4-(2,4-difluorobenz...)
Affinity DataIC50:  46nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310987(CHEMBL1078594 | N-(3-((3-bromo-4-(2,4-difluorobenz...)
Affinity DataIC50:  49nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310986(CHEMBL1078667 | N-(4-((3-chloro-4-(2,4-difluoroben...)
Affinity DataIC50:  55nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310984(3-bromo-4-(2,4-difluorobenzyloxy)-1-(4-((dimethyla...)
Affinity DataIC50:  59nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310983(3-bromo-4-(2,4-difluorobenzyloxy)-1-(3-((dimethyla...)
Affinity DataIC50:  63nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310981(1-(3-(aminomethyl)benzyl)-3-bromo-4-(2,4-difluorob...)
Affinity DataIC50:  65nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310968(4-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  66nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataIC50:  70nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310969(4-((3-chloro-4-(2,4-difluorobenzyloxy)-6-methyl-2-...)
Affinity DataIC50:  79nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310962(3-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  110nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310982(1-(4-(aminomethyl)benzyl)-3-bromo-4-(2,4-difluorob...)
Affinity DataIC50:  120nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310955(3-bromo-4-(2,4-difluorobenzyloxy)-1-(3-fluorobenzy...)
Affinity DataIC50:  130nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310975(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(pyri...)
Affinity DataIC50:  150nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310979(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(2-me...)
Affinity DataIC50:  180nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310963(4-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  190nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310970(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(3-(2...)
Affinity DataIC50:  200nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310976(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(pyri...)
Affinity DataIC50:  210nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310967(3-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  250nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310965(3-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  270nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310973(3-bromo-4-(4-fluorobenzyloxy)-6-methyl-1-(pyridin-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310974(3-bromo-4-(4-fluorobenzyloxy)-6-methyl-1-(pyridin-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310977(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(5-me...)
Affinity DataIC50:  450nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310978(3-bromo-4-(2,4-difluorobenzyloxy)-1-(5-(hydroxymet...)
Affinity DataIC50:  450nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310954(3-bromo-1-(3-fluorobenzyl)-4-(4-fluorobenzyloxy)py...)
Affinity DataIC50:  620nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50318050(1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1H)-one | ...)
Affinity DataIC50:  680nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310951(1-benzyl-4-(benzyloxy)-3-chloropyridin-2(1H)-one |...)
Affinity DataIC50:  900nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310972(3-bromo-4-(4-fluorobenzyloxy)-6-methyl-1-(pyridin-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310961(2-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310980(1-(2-(aminomethyl)benzyl)-3-bromo-4-(2,4-difluorob...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310953(3-bromo-4-(4-chlorobenzyloxy)-1-(4-fluorobenzyl)py...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310964(2-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  2.67E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310952(1-benzyl-4-(benzyloxy)-3-iodopyridin-2(1H)-one | C...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310958(1-benzyl-4-(benzyloxy)-3-methylpyridin-2(1H)-one |...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310957(1-benzyl-4-(benzyloxy)-3-ethylpyridin-2(1H)-one | ...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310960(4-(2,4-difluorobenzyloxy)-1-(3-fluorobenzyl)-2-oxo...)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50240029(1-benzyl-4-(benzyloxy)pyridin-2(1H)-one | CHEMBL26...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310959(4-(benzyloxy)-1-(3-fluorobenzyl)-3-(trifluoromethy...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310956(1-benzyl-4-(benzyloxy)-3-vinylpyridin-2(1H)-one | ...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310965(3-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-o...)
Affinity DataIC50:  1.67E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310984(3-bromo-4-(2,4-difluorobenzyloxy)-1-(4-((dimethyla...)
Affinity DataIC50: >1.71E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50318050(1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1H)-one | ...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310952(1-benzyl-4-(benzyloxy)-3-iodopyridin-2(1H)-one | C...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50240029(1-benzyl-4-(benzyloxy)pyridin-2(1H)-one | CHEMBL26...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310953(3-bromo-4-(4-chlorobenzyloxy)-1-(4-fluorobenzyl)py...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50310954(3-bromo-1-(3-fluorobenzyl)-4-(4-fluorobenzyloxy)py...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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