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Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50030616
TargetAlpha-1B adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataIC50:  0.190nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-1A adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataIC50:  0.254nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2A adrenergic receptor(Human)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50203564((1R,2S,4aR,13bS,14aS)-2-hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataIC50:  3.67nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2C adrenergic receptor(Human)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50203564((1R,2S,4aR,13bS,14aS)-2-hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataIC50:  27.1nMAssay Description:Displacement of radioligand from human adrenergic alpha2C receptor after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-1A adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50:  56nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-1B adrenergic receptor(Rat)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50:  102nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-2A adrenergic receptor(Human)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50299208(4-amino-6-methyl-2-(3-(4-p-tolylpiperazin-1-yl)pro...)
Affinity DataIC50:  320nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed