Compile Data Set for Download or QSAR
maximum 50k data
Found 62 Enz. Inhib. hit(s) with all data for entry = 50030630
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299393(4-((1-benzylpiperidin-4-yl)(3-carbamoylphenyl)amin...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299390(CHEMBL574640 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  0.410nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299385(4-((1-benzylpiperidin-4-yl)(3-hydroxyphenyl)amino)...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299389(4-((1-benzylpiperidin-4-yl)(3-(methylsulfonamido)p...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299382(4-((3-acetylphenyl)(1-benzylpiperidin-4-yl)amino)-...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299388(4-((3-acetamidophenyl)(1-benzylpiperidin-4-yl)amin...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299391(4-((3-aminophenyl)(1-benzylpiperidin-4-yl)amino)-N...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299384(4-((1-benzylpiperidin-4-yl)(3-formylphenyl)amino)-...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299396(4-((1-benzylpiperidin-4-yl)(3-(hydroxymethyl)pheny...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299392(4-((1-benzylpiperidin-4-yl)(3-(methylcarbamoyl)phe...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299386(4-((1-benzylpiperidin-4-yl)(4-carbamoylphenyl)amin...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299395(4-((1-benzylpiperidin-4-yl)(3-((dimethylamino)meth...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299387(4-((1-benzylpiperidin-4-yl)(2-carbamoylphenyl)amin...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299394(CHEMBL575926 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299390(CHEMBL574640 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  75nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299383(4-((1-benzylpiperidin-4-yl)(3-(1-hydroxyethyl)phen...)
Affinity DataKi:  81nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299385(4-((1-benzylpiperidin-4-yl)(3-hydroxyphenyl)amino)...)
Affinity DataKi:  88nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299397(3-((1-benzylpiperidin-4-yl)(4-(diethylcarbamoyl)ph...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299393(4-((1-benzylpiperidin-4-yl)(3-carbamoylphenyl)amin...)
Affinity DataKi:  282nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299399(4-((1-benzylpiperidin-4-yl)(3-((methylamino)methyl...)
Affinity DataKi:  435nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299381(4-((3-(aminomethyl)phenyl)(1-benzylpiperidin-4-yl)...)
Affinity DataKi:  447nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299389(4-((1-benzylpiperidin-4-yl)(3-(methylsulfonamido)p...)
Affinity DataKi:  462nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299386(4-((1-benzylpiperidin-4-yl)(4-carbamoylphenyl)amin...)
Affinity DataKi:  486nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299390(CHEMBL574640 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  576nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299393(4-((1-benzylpiperidin-4-yl)(3-carbamoylphenyl)amin...)
Affinity DataKi:  725nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299385(4-((1-benzylpiperidin-4-yl)(3-hydroxyphenyl)amino)...)
Affinity DataKi:  744nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299381(4-((3-(aminomethyl)phenyl)(1-benzylpiperidin-4-yl)...)
Affinity DataKi:  831nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299388(4-((3-acetamidophenyl)(1-benzylpiperidin-4-yl)amin...)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299384(4-((1-benzylpiperidin-4-yl)(3-formylphenyl)amino)-...)
Affinity DataKi:  1.19E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299398(3-((1-benzylpiperidin-4-yl)(4-(diethylcarbamoyl)ph...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299382(4-((3-acetylphenyl)(1-benzylpiperidin-4-yl)amino)-...)
Affinity DataKi:  1.54E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299395(4-((1-benzylpiperidin-4-yl)(3-((dimethylamino)meth...)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299391(4-((3-aminophenyl)(1-benzylpiperidin-4-yl)amino)-N...)
Affinity DataKi:  2.88E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299381(4-((3-(aminomethyl)phenyl)(1-benzylpiperidin-4-yl)...)
Affinity DataKi:  2.93E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299389(4-((1-benzylpiperidin-4-yl)(3-(methylsulfonamido)p...)
Affinity DataKi:  3.56E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299383(4-((1-benzylpiperidin-4-yl)(3-(1-hydroxyethyl)phen...)
Affinity DataKi:  3.75E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299396(4-((1-benzylpiperidin-4-yl)(3-(hydroxymethyl)pheny...)
Affinity DataKi:  3.81E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299395(4-((1-benzylpiperidin-4-yl)(3-((dimethylamino)meth...)
Affinity DataKi:  4.16E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299391(4-((3-aminophenyl)(1-benzylpiperidin-4-yl)amino)-N...)
Affinity DataKi:  4.25E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299382(4-((3-acetylphenyl)(1-benzylpiperidin-4-yl)amino)-...)
Affinity DataKi:  4.54E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299392(4-((1-benzylpiperidin-4-yl)(3-(methylcarbamoyl)phe...)
Affinity DataKi:  4.71E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299383(4-((1-benzylpiperidin-4-yl)(3-(1-hydroxyethyl)phen...)
Affinity DataKi:  4.74E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299384(4-((1-benzylpiperidin-4-yl)(3-formylphenyl)amino)-...)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299387(4-((1-benzylpiperidin-4-yl)(2-carbamoylphenyl)amin...)
Affinity DataKi:  5.04E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299394(CHEMBL575926 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  5.54E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299386(4-((1-benzylpiperidin-4-yl)(4-carbamoylphenyl)amin...)
Affinity DataKi:  6.18E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299396(4-((1-benzylpiperidin-4-yl)(3-(hydroxymethyl)pheny...)
Affinity DataKi:  6.67E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299394(CHEMBL575926 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  7.10E+3nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299388(4-((3-acetamidophenyl)(1-benzylpiperidin-4-yl)amin...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299387(4-((1-benzylpiperidin-4-yl)(2-carbamoylphenyl)amin...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 62 total ) | Next | Last >>
Jump to: