Compile Data Set for Download or QSAR
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Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50030631
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50040123(CHEMBL438223 | HTry-Gly-Gly-Phe-Leu-Arg-Arg-lle-Ar...)
Affinity DataKi:  1.11nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataKi:  1.85nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299400(CHEMBL584800 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  2.17nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299410(CHEMBL584801 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-D-...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299401(CHEMBL574567 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  3.11nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50040123(CHEMBL438223 | HTry-Gly-Gly-Phe-Leu-Arg-Arg-lle-Ar...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299404(CHEMBL584595 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  3.99nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299402(CHEMBL584799 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  4.56nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299403(CHEMBL584596 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-D-...)
Affinity DataKi:  4.64nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataKi:  6.18nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299405(CHEMBL584594 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  8.17nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50040123(CHEMBL438223 | HTry-Gly-Gly-Phe-Leu-Arg-Arg-lle-Ar...)
Affinity DataKi:  8.18nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50059583(CHEMBL268818 | N-benzyl[D-Pro-10]Dyn A-(1-11) | Ph...)
Affinity DataKi:  14.8nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50002345(CHEMBL407529 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  15.5nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299408(CHEMBL574568 | zyklophin)
Affinity DataKi:  30.3nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299400(CHEMBL584800 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  36.5nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299401(CHEMBL574567 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  44.8nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299402(CHEMBL584799 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  45.1nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299410(CHEMBL584801 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-D-...)
Affinity DataKi:  46.1nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299404(CHEMBL584595 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  49.9nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299403(CHEMBL584596 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-D-...)
Affinity DataKi:  51.2nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50169874((N-alpha-benzyl)Tyr-Gly-Gly-Phe-D-Asn-Arg-Arg-Dap(...)
Affinity DataKi:  66.9nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299405(CHEMBL584594 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  84.9nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50059583(CHEMBL268818 | N-benzyl[D-Pro-10]Dyn A-(1-11) | Ph...)
Affinity DataKi:  98.1nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299400(CHEMBL584800 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299402(CHEMBL584799 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50002345(CHEMBL407529 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299407(CHEMBL574556 | PhCH2Tyr-Gly-Gly-Phe-Leu-D-Asp-Arg-...)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299410(CHEMBL584801 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-D-...)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50059583(CHEMBL268818 | N-benzyl[D-Pro-10]Dyn A-(1-11) | Ph...)
Affinity DataKi:  345nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299404(CHEMBL584595 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  345nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299403(CHEMBL584596 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-D-...)
Affinity DataKi:  372nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299401(CHEMBL574567 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Nalpha...)
Affinity DataKi:  458nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299405(CHEMBL584594 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  474nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50002345(CHEMBL407529 | PhCH2Tyr-Gly-Gly-Phe-Leu-Arg-Arg-ll...)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299407(CHEMBL574556 | PhCH2Tyr-Gly-Gly-Phe-Leu-D-Asp-Arg-...)
Affinity DataKi:  1.19E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299406(CHEMBL585003 | PhCH2Tyr-Gly-Gly-Phe-Leu-D-Asn-Arg-...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50169874((N-alpha-benzyl)Tyr-Gly-Gly-Phe-D-Asn-Arg-Arg-Dap(...)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299406(CHEMBL585003 | PhCH2Tyr-Gly-Gly-Phe-Leu-D-Asn-Arg-...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299407(CHEMBL574556 | PhCH2Tyr-Gly-Gly-Phe-Leu-D-Asp-Arg-...)
Affinity DataKi:  3.66E+3nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299406(CHEMBL585003 | PhCH2Tyr-Gly-Gly-Phe-Leu-D-Asn-Arg-...)
Affinity DataKi:  4.64E+3nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299408(CHEMBL574568 | zyklophin)
Affinity DataKi:  5.88E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50169874((N-alpha-benzyl)Tyr-Gly-Gly-Phe-D-Asn-Arg-Arg-Dap(...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50299408(CHEMBL574568 | zyklophin)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed