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Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50031342
TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311570(2-(6-(4-(4-aminopyrimidin-2-yloxy)piperidin-1-yl)-...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311568(3-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311564(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311569(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311544(2-(2-(1-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)p...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311560(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311556(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311554(2-(1-(6-(2-chlorophenoxy)pyrimidin-4-yl)piperidin-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311551(2-(1-(6-(biphenyl-2-yloxy)pyrimidin-4-yl)piperidin...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311565(5-fluoro-2-(1-(5-fluoro-6-(4-methoxyphenoxy)pyrimi...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311566(3-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311548(5-fluoro-2-(1-(6-(2-methoxyphenoxy)pyrimidin-4-yl)...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311563(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311567(4-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311558(5-fluoro-2-(1-(6-(2-fluorophenoxy)pyrimidin-4-yl)p...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311550(5-fluoro-2-(1-(6-(o-tolyloxy)pyrimidin-4-yl)piperi...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311559(2-(1-(6-(4-chloro-2-methylphenoxy)pyrimidin-4-yl)p...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311562(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311555(2-(1-(6-(2-ethylphenoxy)pyrimidin-4-yl)piperidin-4...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311557(3-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311552(2-(1-(6-(4-chlorophenoxy)pyrimidin-4-yl)piperidin-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311561(2-(6-(4-(4-amino-5-fluoropyrimidin-2-yloxy)piperid...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311549(5-fluoro-2-(1-(6-(p-tolyloxy)pyrimidin-4-yl)piperi...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311553(2-(1-(6-(3-chlorophenoxy)pyrimidin-4-yl)piperidin-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311547(5-fluoro-2-(1-(6-(3-methoxyphenoxy)pyrimidin-4-yl)...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311546(5-fluoro-2-(1-(6-(4-methoxyphenoxy)pyrimidin-4-yl)...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311543(2-((1-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)pip...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311542(2-(1-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)pipe...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311571(2-(6-(4-(4-amino-2-oxopyrimidin-1(2H)-yloxy)piperi...)
Affinity DataIC50:  63nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311545(5-fluoro-2-(1-(6-phenoxypyrimidin-4-yl)piperidin-4...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311541(2-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yloxy)-5-f...)
Affinity DataIC50:  720nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311539(2-(4-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)pipe...)
Affinity DataIC50: >4.00E+3nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311540(2'-deoxy-5-fluorocytidine | 4-amino-5-fluoro-1-((2...)
Affinity DataIC50: >4.00E+3nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB


TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311540(2'-deoxy-5-fluorocytidine | 4-amino-5-fluoro-1-((2...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB


TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311539(2-(4-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)pipe...)
Affinity DataIC50:  5.10E+5nMAssay Description:Inhibition of human dCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311541(2-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yloxy)-5-f...)
Affinity DataEC50:  1.30E+4nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311571(2-(6-(4-(4-amino-2-oxopyrimidin-1(2H)-yloxy)piperi...)
Affinity DataEC50:  350nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311543(2-((1-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)pip...)
Affinity DataEC50:  790nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311544(2-(2-(1-(6-(benzo[b]thiophen-2-yl)pyrimidin-4-yl)p...)
Affinity DataEC50:  160nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311545(5-fluoro-2-(1-(6-phenoxypyrimidin-4-yl)piperidin-4...)
Affinity DataEC50:  340nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311546(5-fluoro-2-(1-(6-(4-methoxyphenoxy)pyrimidin-4-yl)...)
Affinity DataEC50:  890nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311547(5-fluoro-2-(1-(6-(3-methoxyphenoxy)pyrimidin-4-yl)...)
Affinity DataEC50:  36nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311548(5-fluoro-2-(1-(6-(2-methoxyphenoxy)pyrimidin-4-yl)...)
Affinity DataEC50:  17nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311549(5-fluoro-2-(1-(6-(p-tolyloxy)pyrimidin-4-yl)piperi...)
Affinity DataEC50:  60nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311550(5-fluoro-2-(1-(6-(o-tolyloxy)pyrimidin-4-yl)piperi...)
Affinity DataEC50:  19nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311551(2-(1-(6-(biphenyl-2-yloxy)pyrimidin-4-yl)piperidin...)
Affinity DataEC50:  26nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311552(2-(1-(6-(4-chlorophenoxy)pyrimidin-4-yl)piperidin-...)
Affinity DataEC50:  57nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311553(2-(1-(6-(3-chlorophenoxy)pyrimidin-4-yl)piperidin-...)
Affinity DataEC50:  35nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311554(2-(1-(6-(2-chlorophenoxy)pyrimidin-4-yl)piperidin-...)
Affinity DataEC50:  13nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDeoxycytidine kinase(Human)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311555(2-(1-(6-(2-ethylphenoxy)pyrimidin-4-yl)piperidin-4...)
Affinity DataEC50:  61nMAssay Description:Inhibition of dCK in human CCRF-CEM assessed as inhibition of Ara-C phosohorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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