Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50031366
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312032((+/-)-N-(4-(4-methyl-5,6-dihydro-4H-1,3-thiazin-2-...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312033((+/-)-N-(4-(4-isopropyl-5,6-dihydro-4H-1,3-thiazin...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312038((+/-)-N-(4-(4-(4-methoxyphenyl)-5,6-dihydro-4H-1,3...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312037((+/-)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312034((+/-)-N-(4-(4-isobutyl-5,6-dihydro-4H-1,3-thiazin-...)
Affinity DataKi:  62nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312028((+/-)-N-(4-(4-butyl-4,5-dihydrothiazol-2-ylamino)p...)
Affinity DataKi:  69nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312040((+/-)-N-(4-(4-(3-chlorophenyl)-5,6-dihydro-4H-1,3-...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312039((+/-)-N-(4-(4-(4-chlorophenyl)-5,6-dihydro-4H-1,3-...)
Affinity DataKi:  122nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312026((R)-N-(4-(4-ethyl-4,5-dihydrothiazol-2-ylamino)phe...)
Affinity DataKi:  153nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312030((R)-N-(4-(4-phenyl-4,5-dihydrothiazol-2-ylamino)ph...)
Affinity DataKi:  175nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312035((+/-)-N-(4-(4-phenethyl-5,6-dihydro-4H-1,3-thiazin...)
Affinity DataKi:  195nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312017(CHEMBL1082083 | N-(4-(5,6-dihydro-4H-1,3-thiazin-2...)
Affinity DataKi:  221nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312007(CHEMBL1081469 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  248nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312024(5,6-dichloro-N-(4-(5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312020(CHEMBL1080100 | N-(4-(5,6-dihydro-4H-1,3-thiazin-2...)
Affinity DataKi:  318nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312036((+/-)-N-(4-(4-cyclohexyl-5,6-dihydro-4H-1,3-thiazi...)
Affinity DataKi:  332nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312021(6-chloro-N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamin...)
Affinity DataKi:  342nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312025((R)-N-(4-(4-methyl-4,5-dihydrothiazol-2-ylamino)ph...)
Affinity DataKi:  379nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312043((R)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  464nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312027((+/-)-N-(4-(4-propyl-4,5-dihydrothiazol-2-ylamino)...)
Affinity DataKi:  482nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312018(CHEMBL1081181 | N-(4-(5,6-dihydro-4H-1,3-thiazin-2...)
Affinity DataKi:  616nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312029((R)-N-(4-(4-isobutyl-4,5-dihydrothiazol-2-ylamino)...)
Affinity DataKi:  712nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312041((+/-)-N-(4-(4-(2-chlorophenyl)-5,6-dihydro-4H-1,3-...)
Affinity DataKi:  956nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312010(CHEMBL1076207 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312012(CHEMBL1079610 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312013(6-chloro-N-(4-(4,5-dihydrothiazol-2-ylamino)phenet...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312019(CHEMBL1079917 | N-(4-(5,6-dihydro-4H-1,3-thiazin-2...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312011(CHEMBL1079609 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312031(CHEMBL1080289 | N-(4-(5-methoxy-4,5-dihydrothiazol...)
Affinity DataKi:  2.55E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312022(CHEMBL1080102 | N-(4-(5,6-dihydro-4H-1,3-thiazin-2...)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312008(CHEMBL1079440 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  3.46E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312016(5,6-dichloro-N-(4-(4,5-dihydrothiazol-2-ylamino)ph...)
Affinity DataKi:  3.64E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312009(CHEMBL1079441 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  3.99E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312023(CHEMBL1079388 | N-(4-(5,6-dihydro-4H-1,3-thiazin-2...)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312014(CHEMBL1079729 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  5.25E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312015(CHEMBL1079730 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi:  5.92E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 5(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  5.98E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY5 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 5(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312007(CHEMBL1081469 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]pig PPY from human NPY5 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 4(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]human PP from human NPY4 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 4(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312007(CHEMBL1081469 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]human PP from human NPY4 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]pig PPY from human NPY2 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50312007(CHEMBL1081469 | N-(4-(4,5-dihydrothiazol-2-ylamino...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]pig PPY from human NPY2 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed