Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50042293
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423718(CHEMBL606371)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)
Affinity DataIC50:  6.10nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)
Affinity DataIC50:  13nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)
Affinity DataIC50: >20nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)
Affinity DataIC50:  46nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)
Affinity DataIC50:  65nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)
Affinity DataIC50:  79nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)
Affinity DataIC50:  84nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)
Affinity DataIC50:  87nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)
Affinity DataIC50:  100nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)
Affinity DataIC50:  257nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)
Affinity DataIC50:  261nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)
Affinity DataIC50:  319nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)
Affinity DataIC50:  347nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)
Affinity DataIC50:  472nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)
Affinity DataIC50:  502nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423718(CHEMBL606371)
Affinity DataIC50:  703nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)
Affinity DataIC50:  887nMAssay Description:Binding affinity to integrin alpha5beta1 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)
Affinity DataIC50:  890nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)
Affinity DataIC50:  1.34E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)
Affinity DataIC50:  1.60E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)
Affinity DataIC50:  1.73E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)
Affinity DataIC50: >2.00E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423728(CHEMBL593938)
Affinity DataIC50:  2.30E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423721(CHEMBL595105)
Affinity DataIC50:  2.30E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)
Affinity DataIC50:  2.42E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)
Affinity DataIC50:  2.48E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)
Affinity DataIC50:  2.93E+3nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)
Affinity DataIC50:  3.57E+3nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423725(CHEMBL596246)
Affinity DataIC50:  5.20E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423722(CHEMBL593703)
Affinity DataIC50:  7.70E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423726(CHEMBL594161)
Affinity DataIC50:  8.90E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423723(CHEMBL593702)
Affinity DataIC50:  9.70E+3nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423724(CHEMBL596248)
Affinity DataIC50:  1.18E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423727(CHEMBL593226)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to integrin alpha5beta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423720(CHEMBL606866)
Affinity DataIC50:  1.65E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423719(CHEMBL596247)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)
Affinity DataIC50: >5.00E+4nMAssay Description:Binding affinity to integrin alpha2bbeta3 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50423717(CHEMBL594166)
Affinity DataIC50:  9.07E+4nMAssay Description:Binding affinity to integrin alpha5beta5 receptor by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed