Compile Data Set for Download or QSAR
maximum 50k data
Found 136 Enz. Inhib. hit(s) with all data for entry = 50030995
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304973((S)-4-((2-bromobenzyl)(1-(methylsulfonyl)pyrrolidi...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304972((S)-2-chloro-4-((2-chlorobenzyl)(1-(methylsulfonyl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304978((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-chloroben...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304987((S)-4-((2-bromobenzyl)(1-propionylpyrrolidin-3-yl)...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304977((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-methylben...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304975((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-(trifluor...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304976((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-fluoroben...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304964((S)-2-chloro-4-((1-(methylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50:  13nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304957((S)-2-chloro-4-((2-methylbenzyl)(1-propionylpyrrol...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50298028((S)-2-chloro-4-((1-methylpyrrolidin-3-yl)(2-(trifl...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304974((S)-2-chloro-4-((2-methylbenzyl)(1-(methylsulfonyl...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304971((S)-2-chloro-4-((2-fluorobenzyl)(1-(methylsulfonyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304980((S)-methyl 3-((3-chloro-4-cyanophenyl)(5-fluoro-2-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304979((S)-methyl 3-((3-chloro-4-cyanophenyl)(2,3-difluor...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304984((S)-2-chloro-4-((1-propionylpyrrolidin-3-yl)(2-(tr...)
Affinity DataIC50:  25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304985((S)-2-chloro-4-((1-isobutyrylpyrrolidin-3-yl)(2-(t...)
Affinity DataIC50:  25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304958((S)-2-chloro-4-((5-fluoro-2-methylbenzyl)(1-propio...)
Affinity DataIC50:  25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304959((S)-2-chloro-4-((2,5-dichlorobenzyl)(1-propionylpy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304983((S)-4-((1-acetylpyrrolidin-3-yl)(2-(trifluoromethy...)
Affinity DataIC50:  30nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304981((S)-ethyl 3-((3-chloro-4-cyanophenyl)(5-fluoro-2-m...)
Affinity DataIC50:  30nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304961(2-chloro-4-(((S)-1-((S)-2-hydroxypropanoyl)pyrroli...)
Affinity DataIC50:  32nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304965((S)-2-chloro-4-((1-(ethylsulfonyl)pyrrolidin-3-yl)...)
Affinity DataIC50:  40nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304966((S)-2-chloro-4-((1-(isopropylsulfonyl)pyrrolidin-3...)
Affinity DataIC50:  40nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304963(2-chloro-4-((2,5-dichlorobenzyl)((S)-1-((S)-2-hydr...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304986((S)-2-chloro-4-((1-pivaloylpyrrolidin-3-yl)(2-(tri...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304982((S)-isopropyl 3-((3-chloro-4-cyanophenyl)(5-fluoro...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304988((S)-methyl 3-(benzyl(3-chloro-4-cyanophenyl)amino)...)
Affinity DataIC50:  63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304960(2-chloro-4-(((S)-1-((S)-2-hydroxypropanoyl)pyrroli...)
Affinity DataIC50:  63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304990((S)-4-((1-(butylsulfonyl)pyrrolidin-3-yl)(2-(trifl...)
Affinity DataIC50:  63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304969((S)-4-(benzyl(1-(methylsulfonyl)pyrrolidin-3-yl)am...)
Affinity DataIC50:  63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304962(2-chloro-4-((5-fluoro-2-methylbenzyl)((S)-1-((S)-2...)
Affinity DataIC50:  79nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304968((S)-2-chloro-4-((1-(isobutylsulfonyl)pyrrolidin-3-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304967((S)-2-chloro-4-((1-(propylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50:  80nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304989((S)-2-chloro-4-((1-(methylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50:  100nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304970((S)-2-chloro-4-((2-cyanobenzyl)(1-(methylsulfonyl)...)
Affinity DataIC50:  100nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304967((S)-2-chloro-4-((1-(propylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50:  110nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304968((S)-2-chloro-4-((1-(isobutylsulfonyl)pyrrolidin-3-...)
Affinity DataIC50:  160nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304975((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-(trifluor...)
Affinity DataIC50:  160nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304966((S)-2-chloro-4-((1-(isopropylsulfonyl)pyrrolidin-3...)
Affinity DataIC50:  280nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304964((S)-2-chloro-4-((1-(methylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50:  330nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304965((S)-2-chloro-4-((1-(ethylsulfonyl)pyrrolidin-3-yl)...)
Affinity DataIC50:  350nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304986((S)-2-chloro-4-((1-pivaloylpyrrolidin-3-yl)(2-(tri...)
Affinity DataIC50:  440nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304977((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-methylben...)
Affinity DataIC50:  680nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304973((S)-4-((2-bromobenzyl)(1-(methylsulfonyl)pyrrolidi...)
Affinity DataIC50:  690nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304985((S)-2-chloro-4-((1-isobutyrylpyrrolidin-3-yl)(2-(t...)
Affinity DataIC50:  720nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50298028((S)-2-chloro-4-((1-methylpyrrolidin-3-yl)(2-(trifl...)
Affinity DataIC50:  780nMAssay Description:Inhibition of human ERG by patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304972((S)-2-chloro-4-((2-chlorobenzyl)(1-(methylsulfonyl...)
Affinity DataIC50:  870nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304978((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-chloroben...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50298028((S)-2-chloro-4-((1-methylpyrrolidin-3-yl)(2-(trifl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304982((S)-isopropyl 3-((3-chloro-4-cyanophenyl)(5-fluoro...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 136 total ) | Next | Last >>
Jump to: