Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50004267
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12216BDBM12216((2R,3R,4R,5R)-2,5-bis(benzyloxy)-3,4-dihydroxy-N-[...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12216BDBM12216((2R,3R,4R,5R)-2,5-bis(benzyloxy)-3,4-dihydroxy-N-[...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480920BDBM50480920(CHEMBL367384)
Affinity DataKi:  0.600nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480923BDBM50480923(CHEMBL573789)
Affinity DataKi:  2.30nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480928BDBM50480928(CHEMBL573868)
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480924BDBM50480924(CHEMBL573717)
Affinity DataKi:  700nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480921BDBM50480921(CHEMBL573845)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480922BDBM50480922(CHEMBL573809)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480927BDBM50480927(CHEMBL573888)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480926BDBM50480926(CHEMBL573849)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Stockholm University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480925BDBM50480925(CHEMBL584774)
Affinity DataKi:  9.90E+4nMAssay Description:Inhibition of HIV1 recombinant protease by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed