Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50004317
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481575BDBM50481575(CHEMBL591351)
Affinity DataIC50: 6.14E+3nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481577BDBM50481577(CHEMBL591596)
Affinity DataIC50: 2.88E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481573BDBM50481573(CHEMBL591295)
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481574BDBM50481574(CHEMBL589855)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481576BDBM50481576(CHEMBL589658)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481570BDBM50481570(CHEMBL589505)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481571BDBM50481571(CHEMBL591595)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481572BDBM50481572(CHEMBL589905)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated NotchdeltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed