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Found 15 Enz. Inhib. hit(s) with all data for entry = 50031220
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  185nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)
Affinity DataIC50:  350nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  375nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309173((1S,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  425nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309174((1S,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  548nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309173((1S,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  825nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309174((1S,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309174((1S,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309173((1S,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute Of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed