Affinity DataKi: 1.29nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.31nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.38nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 3.59nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.17nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.41nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 6.04nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 13.7nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 14.4nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 27.3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 38.8nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 171nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 248nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia
Curated by ChEMBL
University Of Pavia
Curated by ChEMBL
Affinity DataKi: 841nMAssay Description:Displacement of [3H]-U-69593 from kappa-type opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair