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Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50039083
TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)
Affinity DataKi:  17nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50201010(((2R,3aR,4R,6R,6aR)-4-(hydroxymethyl)-6-(5-methyl-...)
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50310202((2-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-...)
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50310201((1-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-...)
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50310199((1-fluoro-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimid...)
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50310200((1-hydroxy-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimi...)
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50310203(8-(5-bromo-3-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydro...)
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378690(CHEMBL597306)
Affinity DataIC50:  11nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378691(CHEMBL609919)
Affinity DataIC50:  15nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378689(CHEMBL599563)
Affinity DataIC50:  45nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378684(CHEMBL599543)
Affinity DataIC50:  45nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378687(CHEMBL598328)
Affinity DataIC50:  190nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378688(CHEMBL599562)
Affinity DataIC50:  220nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378685(CHEMBL599544)
Affinity DataIC50:  250nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378692(CHEMBL611383)
Affinity DataIC50:  300nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378686(CHEMBL598327)
Affinity DataIC50:  350nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThymidine phosphorylase(Rat)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378683(CHEMBL599132)
Affinity DataIC50:  750nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed