Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50039012
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378570(CHEMBL572085)
Affinity DataIC50:  24nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378570(CHEMBL572085)
Affinity DataIC50:  180nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378570(CHEMBL572085)
Affinity DataIC50:  240nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378569(CHEMBL570324)
Affinity DataIC50:  520nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378575(CHEMBL571845)
Affinity DataIC50:  920nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378575(CHEMBL571845)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378571(CHEMBL572293)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378575(CHEMBL571845)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378571(CHEMBL572293)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378571(CHEMBL572293)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50237601(CHEMBL411941 | CycloRGDfV | [(2S,5R,8S,11S)-5-Benz...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50237601(CHEMBL411941 | CycloRGDfV | [(2S,5R,8S,11S)-5-Benz...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378569(CHEMBL570324)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378569(CHEMBL570324)
Affinity DataIC50:  2.52E+4nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50237601(CHEMBL411941 | CycloRGDfV | [(2S,5R,8S,11S)-5-Benz...)
Affinity DataIC50:  3.47E+4nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378577(CHEMBL571979)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378576(CHEMBL570087)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378574(CHEMBL571628)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378573(CHEMBL572266)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378572(CHEMBL570963)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378577(CHEMBL571979)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378576(CHEMBL570087)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378573(CHEMBL572266)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378572(CHEMBL570963)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378577(CHEMBL571979)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378576(CHEMBL570087)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378574(CHEMBL571628)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378573(CHEMBL572266)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378572(CHEMBL570963)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50378574(CHEMBL571628)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed