Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50039012
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378570BDBM50378570(CHEMBL572085)
Affinity DataIC50: 24nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378570BDBM50378570(CHEMBL572085)
Affinity DataIC50: 180nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378570BDBM50378570(CHEMBL572085)
Affinity DataIC50: 240nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378569BDBM50378569(CHEMBL570324)
Affinity DataIC50: 520nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378575BDBM50378575(CHEMBL571845)
Affinity DataIC50: 920nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378575BDBM50378575(CHEMBL571845)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378571BDBM50378571(CHEMBL572293)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378575BDBM50378575(CHEMBL571845)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378571BDBM50378571(CHEMBL572293)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378571BDBM50378571(CHEMBL572293)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50237601BDBM50237601([5-Benzyl-11-(3-guanidino-propyl)-8-isopropyl-3,6,...)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50237601BDBM50237601([5-Benzyl-11-(3-guanidino-propyl)-8-isopropyl-3,6,...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378569BDBM50378569(CHEMBL570324)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378569BDBM50378569(CHEMBL570324)
Affinity DataIC50: 2.52E+4nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50237601BDBM50237601([5-Benzyl-11-(3-guanidino-propyl)-8-isopropyl-3,6,...)
Affinity DataIC50: 3.47E+4nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378576BDBM50378576(CHEMBL570087)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378574BDBM50378574(CHEMBL571628)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378577BDBM50378577(CHEMBL571979)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378572BDBM50378572(CHEMBL570963)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378573BDBM50378573(CHEMBL572266)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in human SK-MEL-24 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378574BDBM50378574(CHEMBL571628)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378576BDBM50378576(CHEMBL570087)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378577BDBM50378577(CHEMBL571979)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378574BDBM50378574(CHEMBL571628)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378572BDBM50378572(CHEMBL570963)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378573BDBM50378573(CHEMBL572266)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378577BDBM50378577(CHEMBL571979)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378572BDBM50378572(CHEMBL570963)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378576BDBM50378576(CHEMBL570087)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alphavbeta3 integrin-mediated cell adhesion in HUVEC on vitronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378573BDBM50378573(CHEMBL572266)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of alpha5beta1 integrin-mediated cell adhesion in human K562 cells on fibronectin coated plate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed