Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50031272
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  33nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310276(CHEMBL601625 | N-Hexadecyl 2-(5-hydroxy-4-oxo-2-ph...)
Affinity DataIC50:  35nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310266(CHEMBL598307 | Hexadecyl 2-(5-hydroxy-4-oxo-2-phen...)
Affinity DataIC50:  48nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310275(CHEMBL598520 | N-Tetradecyl 2-(5-hydroxy-4-oxo-2-p...)
Affinity DataIC50:  316nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310257(CHEMBL600381 | N-Octadecyl 2-(5-hydroxy-4-oxo-2-ph...)
Affinity DataIC50:  464nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310267(CHEMBL597096 | Octadecyl 2-(5-hydroxy-4-oxo-2-phen...)
Affinity DataIC50:  692nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310265(CHEMBL598306 | Tetradecyl 2-(5-hydroxy-4-oxo-2-phe...)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310274(CHEMBL597914 | N-Dodecyl 2-(5-hydroxy-4-oxo-2-phen...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310258(CHEMBL592153 | N-Icosyl 2-(5-hydroxy-4-oxo-2-pheny...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310268(CHEMBL591495 | Icosyl 2-(5-hydroxy-4-oxo-2-phenyl-...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310264(CHEMBL598305 | Dodecyl 2-(5-hydroxy-4-oxo-2-phenyl...)
Affinity DataIC50:  1.72E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310273(CHEMBL605337 | N-Decyl 2-(5-hydroxy-4-oxo-2-phenyl...)
Affinity DataIC50:  2.14E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310263(CHEMBL599728 | Decyl 2-(5-hydroxy-4-oxo-2-phenyl-4...)
Affinity DataIC50:  3.11E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310272(CHEMBL597708 | N-Nonyl 2-(5-hydroxy-4-oxo-2-phenyl...)
Affinity DataIC50:  3.58E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310262(CHEMBL599145 | Nonyl 2-(5-hydroxy-4-oxo-2-phenyl-4...)
Affinity DataIC50:  4.96E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310271(CHEMBL597304 | N-Octyl 2-(5-hydroxy-4-oxo-2-phenyl...)
Affinity DataIC50:  5.33E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310261(CHEMBL603968 | Octyl 2-(5-hydroxy-4-oxo-2-phenyl-4...)
Affinity DataIC50:  5.84E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310270(CHEMBL597303 | N-Heptyl 2-(5-hydroxy-4-oxo-2-pheny...)
Affinity DataIC50:  6.28E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310260(CHEMBL599524 | Heptyl 2-(5-hydroxy-4-oxo-2-phenyl-...)
Affinity DataIC50:  7.23E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310269(CHEMBL611681 | N-Hexyl-2-(5-hydroxy-4-oxo-2-phenyl...)
Affinity DataIC50:  8.71E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50310259(CHEMBL591213 | Hexyl 2-(5-hydroxy-4-oxo-2-phenyl-4...)
Affinity DataIC50:  9.12E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed