Compile Data Set for Download or QSAR
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Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50031066
TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306358(5-(4-(3,5-dimethylphenoxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  96nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306360(5-(4-(2,4-dimethylphenoxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  121nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306361(5-(4-(2,5-dimethylphenoxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  238nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306362(5-(4-(3,4-dimethylphenoxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  727nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306363(5-(4-(2-chlorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  1.19E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306364(5-(4-(3-chlorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  318nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306365(5-(4-(4-chlorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306366(5-(4-(3,5-dichlorophenoxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  207nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306367(5-(4-(2-chloro-4-(trifluoromethyl)phenoxy)benzyl)t...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306368(4-(4-((2,4-dioxothiazolidin-5-yl)methyl)phenoxy)-2...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306369(5-(4-(naphthalen-1-yloxy)benzyl)thiazolidine-2,4-d...)
Affinity DataEC50:  135nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306370(5-(4-(3-(trifluoromethyl)pyridin-2-yloxy)benzyl)th...)
Affinity DataEC50:  2.29E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306371(5-(4-(4-(trifluoromethyl)pyridin-2-yloxy)benzyl)th...)
Affinity DataEC50:  237nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306372(5-(4-(5-(trifluoromethyl)pyridin-2-yloxy)benzyl)th...)
Affinity DataEC50:  558nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306373(5-(4-(6-(trifluoromethyl)pyridin-2-yloxy)benzyl)th...)
Affinity DataEC50:  1.64E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306374(5-(4-(3-methylpyridin-2-yloxy)benzyl)thiazolidine-...)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306375(5-(4-(4-methylpyridin-2-yloxy)benzyl)thiazolidine-...)
Affinity DataEC50:  4.28E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306376(5-(4-(5-methylpyridin-2-yloxy)benzyl)thiazolidine-...)
Affinity DataEC50:  4.47E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306377(5-(4-(6-methylpyridin-2-yloxy)benzyl)thiazolidine-...)
Affinity DataEC50:  2.62E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306378(5-(4-(5-chloropyridin-2-yloxy)benzyl)thiazolidine-...)
Affinity DataEC50:  1.87E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306379(5-(4-(6-methyl-4-(trifluoromethyl)pyridin-2-yloxy)...)
Affinity DataEC50:  218nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306380(5-(4-(4-methyl-6-(trifluoromethyl)pyridin-2-yloxy)...)
Affinity DataEC50:  688nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306381(5-(4-(3-chloro-5-(trifluoromethyl)pyridin-2-yloxy)...)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306382(5-(4-(3,5-dichloropyridin-2-yloxy)benzyl)thiazolid...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306383(5-(4-(isoquinolin-3-yloxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  144nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306384(5-(4-(3-chloro-5-(trifluoromethyl)pyridin-2-yloxy)...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306385(5-(4-(2-chloro-4-(trifluoromethyl)phenoxy)-2-methy...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306386(5-(2-chloro-4-(3-chloro-5-(trifluoromethyl)pyridin...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306387(5-(2-chloro-4-(3,5-dichloropyridin-2-yloxy)benzyl)...)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306388(5-(4-(2,4-dichlorophenoxy)-2-(trifluoromethyl)benz...)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306389(5-(4-(2,4-dichlorophenoxy)-2-methoxybenzyl)thiazol...)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306390(5-(4-(3-chloro-5-(trifluoromethyl)pyridin-2-yloxy)...)
Affinity DataEC50:  1.39E+4nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306391(5-(4-(3-chloro-5-(trifluoromethyl)pyridin-2-yloxy)...)
Affinity DataEC50:  5.45E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306392(5-((4-(3-chloro-5-(trifluoromethyl)pyridin-2-yloxy...)
Affinity DataEC50:  2.36E+4nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306393(5-(4-(4-fluorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306394(5-(4-(2,4-dichlorophenoxy)benzyl)thiazolidine-2,4-...)
Affinity DataEC50:  101nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306395(5-(4-(2,4-dichlorophenoxy)benzyl)oxazolidine-2,4-d...)
Affinity DataEC50:  4.02E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306396(3-(4-(2,4-dichlorophenoxy)benzyl)pyrrolidine-2,5-d...)
Affinity DataEC50:  6.45E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306397(5-(4-phenoxybenzyl)thiazolidine-2,4-dione | CHEMBL...)
Affinity DataEC50:  307nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306398(5-(3-phenoxybenzyl)thiazolidine-2,4-dione | CHEMBL...)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306399(5-(2-phenoxybenzyl)thiazolidine-2,4-dione | CHEMBL...)
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306400(5-(4-(phenylthio)benzyl)thiazolidine-2,4-dione | C...)
Affinity DataEC50:  5.06E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306401(5-(4-benzylbenzyl)thiazolidine-2,4-dione | CHEMBL5...)
Affinity DataEC50:  9.28E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306402(5-(4-styrylbenzyl)thiazolidine-2,4-dione | CHEMBL5...)
Affinity DataEC50:  2.09E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306403(5-(4-phenethylbenzyl)thiazolidine-2,4-dione | CHEM...)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145471(5-(4-(benzyloxy)benzyl)thiazolidine-2,4-dione | 5-...)
Affinity DataEC50:  6.18E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306404(5-(4-benzoylbenzyl)thiazolidine-2,4-dione | CHEMBL...)
Affinity DataEC50:  5.30E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306405(5-(biphenyl-4-ylmethyl)thiazolidine-2,4-dione | CH...)
Affinity DataEC50:  2.22E+3nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFree fatty acid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50306406(5-(4-(o-tolyloxy)benzyl)thiazolidine-2,4-dione | C...)
Affinity DataEC50:  124nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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