Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50030917
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304008(3-(4-Fluorophenyl)-2-(2-isopropylaminopyridin-4-yl...)
Affinity DataIC50:  38nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304016(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-isopropylp...)
Affinity DataIC50:  81nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304010(CHEMBL567260 | N-sec-Butyl-4-(3-(4-fluorophenyl)qu...)
Affinity DataIC50:  114nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304013(4-(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)pyridin-2-...)
Affinity DataIC50:  211nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304009(4-(3-(4-Fluorophenyl)-6,7-dimethylquinoxalin-2-yl)...)
Affinity DataIC50:  238nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304017(4-(4-(3-(4-Fluorophenyl)-6,7-dimethylquinoxalin-2-...)
Affinity DataIC50:  259nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  290nMAssay Description:Inhibition of JNK3 by nonradioactive JNK3 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304011(2-(4-Fluorophenyl)-3-(2-isopropylaminopyridin-4-yl...)
Affinity DataIC50:  333nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304014(4-(6,7-Dichlor-3-(4-fluorophenyl)quinoxalin-2-yl)-...)
Affinity DataIC50:  412nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304015(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-((S)-1-phe...)
Affinity DataIC50:  431nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304012(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-((S)-3-met...)
Affinity DataIC50:  576nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304021(CHEMBL566205 | N-sec-Butyl-4-(3-(4-fluorophenyl)-6...)
Affinity DataIC50:  595nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304018(4-(4-(6,7-Dichloro-3-(4-fluorophenyl)quinoxalin-2-...)
Affinity DataIC50:  608nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304029(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-isobutylpy...)
Affinity DataIC50:  642nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304015(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-((S)-1-phe...)
Affinity DataIC50:  720nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304012(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-((S)-3-met...)
Affinity DataIC50:  790nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304020(4-(3-(4-Fluorophenyl)-6,7-dimethylquinoxalin-2-yl)...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304022(CHEMBL565385 | N-Benzyl-4-(3-(4-fluorophenyl)-6,7-...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304024(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-((R)-3-met...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304025(2-(4-Fluorophenyl)-3-(pyridin-4-yl)quinoxaline | C...)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304023(3-(4-Fluorophenyl)-2-(pyridin-4-yl)pyrido[2,3-b]py...)
Affinity DataIC50:  3.19E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304026(2-(4-Fluorophenyl)-6,7-dimethyl-3-(pyridin-4-yl)qu...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304016(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-isopropylp...)
Affinity DataIC50:  3.95E+3nMAssay Description:Inhibition of JNK3 by nonradioactive JNK3 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304019(4-(3-(4-Fluorophenyl)quinoxalin-2-yl)-N-((R)-1-phe...)
Affinity DataIC50:  4.79E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304027(3-(4-Fluorophenyl)-6-methoxy-2-(pyridin-4-yl)quino...)
Affinity DataIC50:  6.14E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304028(4-(6,7-Dichloro-3-(4-fluorophenyl)quinoxalin-2-yl)...)
Affinity DataIC50:  9.46E+3nMAssay Description:Inhibition of p38alpha-mediated ATF2 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard-Karls-University Of T£Bingen

Curated by ChEMBL
LigandPNGBDBM50304025(2-(4-Fluorophenyl)-3-(pyridin-4-yl)quinoxaline | C...)
Affinity DataIC50:  3.18E+4nMAssay Description:Inhibition of JNK3 by nonradioactive JNK3 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed