Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50035947
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421887BDBM50421887(CHEMBL2112181)
Affinity DataEC50:  5.40nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25400BDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataEC50:  12.6nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50367678BDBM50367678(CHEMBL605469)
Affinity DataEC50:  33.9nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  63.1nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009525BDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataEC50:  191nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82031BDBM82031(CAS_1818-71-9 | isoguanosine | 2-Oxoado (isoguanos...)
Affinity DataEC50:  1.15E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368251BDBM50368251(CHEMBL605879)
Affinity DataEC50:  2.19E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368264BDBM50368264(CHEMBL603588)
Affinity DataEC50:  2.63E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 14487BDBM14487([U-14C]adenosine | CHEMBL477 | cid_60961 | (2R,3R,...)
Affinity DataEC50:  3.39E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368250BDBM50368250(CHEMBL605254)
Affinity DataEC50:  3.72E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368253BDBM50368253(CHEMBL603373)
Affinity DataEC50:  4.47E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50364062BDBM50364062(CHEMBL1950555)
Affinity DataEC50:  5.62E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368258BDBM50368258(CHEMBL606093)
Affinity DataEC50:  8.71E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368261BDBM50368261(CHEMBL605247)
Affinity DataEC50:  8.71E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421888BDBM50421888(CHEMBL2311198)
Affinity DataEC50:  9.33E+3nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataEC50:  1.26E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368243BDBM50368243(CHEMBL605466)
Affinity DataEC50:  1.38E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368242BDBM50368242(CHEMBL603589)
Affinity DataEC50:  1.41E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368262BDBM50368262(CHEMBL604429)
Affinity DataEC50:  1.59E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368263BDBM50368263(CHEMBL604223)
Affinity DataEC50:  2.29E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 35804BDBM35804(3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl...)
Affinity DataEC50:  2.46E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368245BDBM50368245(CHEMBL604009)
Affinity DataEC50:  3.55E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368244BDBM50368244(CHEMBL603379)
Affinity DataEC50:  3.72E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368254BDBM50368254(CHEMBL605464)
Affinity DataEC50:  4.57E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368259BDBM50368259(CHEMBL605673)
Affinity DataEC50:  5.01E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368256BDBM50368256(CHEMBL603374)
Affinity DataEC50:  6.31E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368246BDBM50368246(CHEMBL604224)
Affinity DataEC50:  6.61E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368255BDBM50368255(CHEMBL604844)
Affinity DataEC50:  7.94E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421886BDBM50421886(CHEMBL2311200)
Affinity DataEC50:  7.94E+4nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368248BDBM50368248(CHEMBL605472)
Affinity DataEC50:  1.00E+5nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368247BDBM50368247(CHEMBL604838)
Affinity DataEC50:  1.07E+5nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368260BDBM50368260(CHEMBL606510)
Affinity DataEC50:  1.48E+5nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368265BDBM50368265(CHEMBL604426)
Affinity DataEC50:  2.24E+5nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368249BDBM50368249(CHEMBL605679)
Affinity DataEC50:  8.91E+5nMAssay Description:Prolongation of the stimulus-QRS interval by 50% of the maximum response at the Adenosine A1 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed