Affinity DataIC50: 3.68E+3nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]bombesin from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation counti...More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]bombesin from human bombesin BB2 receptor expressed in NFAT-CHO cells after 2 hrs by liquid sci...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]bombesin from human bombesin BB1 receptor expressed in NFAT-CHO cells after 2 hrs by liquid sci...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 174nMAssay Description:Agonistic activity at rat BRS3 expressed in HEK293AEO at 10 uM by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 238nMAssay Description:Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.66E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.18E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.72E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.76E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.62E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.71E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.38E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.95E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 205nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.32E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.72E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.12E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.36E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.48E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 812nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.89E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 127nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.31E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.66E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 292nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 825nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.29E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 177nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 159nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 588nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 133nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 41nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 88nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 642nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 375nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 338nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 119nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 106nMAssay Description:Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 527nMAssay Description:Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 165nMAssay Description:Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 340nMAssay Description:Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 184nMAssay Description:Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.24E+3nMAssay Description:Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair