Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50039065
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM20880((2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)me...)
Affinity DataIC50:  0.490nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308460((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-3-yl)...)
Affinity DataIC50:  3.51nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308448(2-(2-Chloro-5-((2S,3S,4R,5R,6R)-3,4,5-tris(benzylo...)
Affinity DataIC50:  4.06nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM20878((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-{2-[(4-methox...)
Affinity DataIC50:  6.25nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308450((2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)-1,...)
Affinity DataIC50:  7.03nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308454((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-phenylfuran-...)
Affinity DataIC50:  10.6nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308436((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(methylthio)-1,...)
Affinity DataIC50:  10.9nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308459((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-2-yl)...)
Affinity DataIC50:  14.4nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308440((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-phenyl-1,3,4-th...)
Affinity DataIC50:  16.6nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308451((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-3-yl)-1,...)
Affinity DataIC50:  17.7nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308463((2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(5-chlorothioph...)
Affinity DataIC50:  18.2nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308465((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiazol-4-yl)-...)
Affinity DataIC50:  21.8nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308476((3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-propylphenyl)-1...)
Affinity DataIC50:  24.9nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308442((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pyridin-2-yl)-...)
Affinity DataIC50:  30.3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308445((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-methylpyridi...)
Affinity DataIC50:  36.4nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308464((2S,3R,4R,5S,6R)-2-(3-((5-(Benzo[b]thiophen-2-yl)-...)
Affinity DataIC50:  44.5nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308477((3R,4R,5S,6R)-2-(4-chloro-3-((5-(pyridin-3-yl)-1,3...)
Affinity DataIC50:  45.3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308478((3R,4R,5S,6R)-2-(4-chloro-3-((5-(pyridin-4-yl)-1,3...)
Affinity DataIC50:  53nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308453((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-methylfuran-...)
Affinity DataIC50:  58.3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308466(((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-(pyridin-4-...)
Affinity DataIC50:  72.6nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308446((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(isoquinolin-3-...)
Affinity DataIC50:  81.6nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308444((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(6-methylpyridi...)
Affinity DataIC50:  97.4nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308475((3R,4R,5S,6R)-2-(4-Chloro-3-((5-p-tolyl-1,3,4-thia...)
Affinity DataIC50:  103nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308452((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-methylfuran-...)
Affinity DataIC50:  106nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308457(((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(1-methyl-1Hpy...)
Affinity DataIC50:  119nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308484((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-heptyl-1,3,4-th...)
Affinity DataIC50:  122nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308441((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-chlorophenyl...)
Affinity DataIC50:  126nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308435((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-methoxy-1,3,4-t...)
Affinity DataIC50:  146nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308437((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(trifluoromethy...)
Affinity DataIC50:  155nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308449((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pyridazin-4-yl...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308481((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-propyl-1,3,4-th...)
Affinity DataIC50:  214nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308455((2S,3R,4R,5S,6R)-2-(3-((5-(Benzofuran-2-yl)-1,3,4-...)
Affinity DataIC50:  249nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308456((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-methylisoxaz...)
Affinity DataIC50:  257nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308483((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-pentyl-1,3,4-th...)
Affinity DataIC50:  353nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308482((2S,3R,4R,5S,6R)-2-(3-((5-Butyl-1,3,4-thiadiazol-2...)
Affinity DataIC50:  379nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308439((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-cyclopentyl-1,3...)
Affinity DataIC50:  445nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308474((3R,4R,5S,6R)-2-(4-Chloro-3-((5-cyclohexyl-1,3,4-t...)
Affinity DataIC50:  542nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308447(((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(quinolin-2-yl...)
Affinity DataIC50:  562nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308443((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(6-methylpyridi...)
Affinity DataIC50:  638nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308462((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-chlorothioph...)
Affinity DataIC50:  712nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308438((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2,2,2-trifluor...)
Affinity DataIC50:  758nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308461((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-methylthioph...)
Affinity DataIC50:  762nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308473((2R,3S,4R,5R)-2-(Hydroxymethyl)-6-(3-((5-(pyridin-...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308472((2R,3S,4R,5R)-2-(Hydroxymethyl)-6-(3-((5-phenyl-1,...)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308479((3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-chlorobenzyl)-1...)
Affinity DataIC50:  2.39E+3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308458((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(1-methyl-1Hind...)
Affinity DataIC50:  3.28E+3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308470((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-2-yl)-1,...)
Affinity DataIC50:  6.91E+3nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308480((3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-(4-chlorophenyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308468(((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-ethyl-5-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50308467((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3,5-dimethylis...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant SGLT2 expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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