Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50004350
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482057BDBM50482057(CHEMBL1092328)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482058BDBM50482058(CHEMBL1091563)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482059BDBM50482059(CHEMBL1093188)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482060BDBM50482060(CHEMBL1089200)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482062BDBM50482062(CHEMBL1091494)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482061BDBM50482061(CHEMBL1089530)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482056BDBM50482056(CHEMBL1092725)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of gamma-secretase-mediated Notch deltaE cleavage in human HeLa cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed