Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50035958
TargetSodium-dependent dopamine transporter(Rat)
Research Biochemicals

Curated by ChEMBL
LigandPNGBDBM50451132(WIN-35428 | CHEMBL2079586)
Affinity DataIC50: 18nMAssay Description:Compound was evaluated for inhibition of specifically bound [3H]- cocaine (2.7 nM) against Dopamine transporter in cynomolgus monkeysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Research Biochemicals

Curated by ChEMBL
LigandPNGBDBM50005550(CHEMBL48225 | 8-Allyl-3-(4-fluoro-phenyl)-8-aza-bi...)
Affinity DataIC50: 23nMAssay Description:Compound was evaluated for inhibition of specifically bound [3H]- cocaine (2.7 nM) against Dopamine transporter in cynomolgus monkeysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Research Biochemicals

Curated by ChEMBL
LigandPNGBDBM50012154(CHEMBL21112 | 3-(4-Fluoro-phenyl)-8-aza-bicyclo[3....)
Affinity DataIC50: 36nMAssay Description:Compound was evaluated for inhibition of specifically bound [3H]- cocaine (2.7 nM) against Dopamine transporter in cynomolgus monkeysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Research Biochemicals

Curated by ChEMBL
LigandPNGBDBM50005542(CHEMBL416818 | 3-(4-Fluoro-phenyl)-8-propyl-8-aza-...)
Affinity DataIC50: 43nMAssay Description:Compound was evaluated for inhibition of specifically bound [3H]- cocaine (2.7 nM) against Dopamine transporter in cynomolgus monkeysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Research Biochemicals

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataIC50: 68nMAssay Description:Compound was evaluated for inhibition of specifically bound [3H]- cocaine (2.7 nM) against Dopamine transporter in cynomolgus monkeysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed