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Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50039145
TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317448(7-Benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-...)
Affinity DataEC50:  380nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317449(7-benzyl-5-(pyrrolidin-1-yl)-6,7,8,9-tetrahydro-3H...)
Affinity DataEC50:  965nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317450(5-(azepan-1-yl)-7-benzyl-6,7,8,9-tetrahydro-3H-pyr...)
Affinity DataEC50:  1.44E+3nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317443(1-(1-amino-7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tet...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317444(7-benzyl-3-methyl-5-(piperidin-1-yl)-6,7,8,9-tetra...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317445(7-benzyl-N-neopentyl-5-(piperidin-1-yl)-6,7,8,9-te...)
Affinity DataEC50:  4.15E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317446(7-benzyl-N-ethyl-5-(piperidin-1-yl)-6,7,8,9-tetrah...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317447(CHEMBL1099135 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  543nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317451(CHEMBL1098838 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  704nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317452(CHEMBL1098837 | N-(7-Benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317453(CHEMBL1098836 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  1.54E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317454(CHEMBL1096193 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  4.76E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317455(CHEMBL1099123 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  3.47E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317456(CHEMBL1099122 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317457(7-(4-Fluorobenzoyl)-5-(piperidin-1-yl)-6,7,8,9-tet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317458(7-phenethyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317459(7-neopentyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317460(7-isobutyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317461(7-(cyclohexylmethyl)-5-(piperidin-1-yl)-6,7,8,9-te...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317462(7-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(piperidin-1-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317463(5-(piperidin-1-yl)-7-(3-(trifluoromethyl)benzyl)-6...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317464(7-(4-methoxybenzyl)-5-(piperidin-1-yl)-6,7,8,9-tet...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317466(7-(2-chlorobenzyl)-5-(piperidin-1-yl)-6,7,8,9-tetr...)
Affinity DataEC50:  5.57E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317467(5-(Piperidin-1-yl)-7-(pyridin-2-ylmethyl)-6,7,8,9-...)
Affinity DataEC50:  6.78E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50378777(CHEMBL1204083)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317469(7-benzyl-N5-phenyl-6,7,8,9-tetrahydro-3H-pyrazolo[...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317470(7-benzyl-N5-cyclohexyl-6,7,8,9-tetrahydro-3H-pyraz...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317471(7-benzyl-N5-isopropyl-6,7,8,9-tetrahydro-3H-pyrazo...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317472(7-benzyl-N5,N5-dimethyl-6,7,8,9-tetrahydro-3H-pyra...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317473(7-benzyl-5-(4-methylpiperazin-1-yl)-6,7,8,9-tetrah...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317474(7-benzyl-5-(piperazin-1-yl)-6,7,8,9-tetrahydro-3H-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317475(7-benzyl-5-morpholino-6,7,8,9-tetrahydro-3H-pyrazo...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317476(7-benzyl-5-(4-fluoropiperidin-1-yl)-6,7,8,9-tetrah...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317477(7-benzyl-5-(4-methylpiperidin-1-yl)-6,7,8,9-tetrah...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317478(5-(azocan-1-yl)-7-benzyl-6,7,8,9-tetrahydro-3H-pyr...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317450(5-(azepan-1-yl)-7-benzyl-6,7,8,9-tetrahydro-3H-pyr...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317449(7-benzyl-5-(pyrrolidin-1-yl)-6,7,8,9-tetrahydro-3H...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50317448(7-Benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-...)
Affinity DataEC50:  4.53E+3nMAssay Description:Agonist activity at human BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317443(1-(1-amino-7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tet...)
Affinity DataEC50:  759nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317444(7-benzyl-3-methyl-5-(piperidin-1-yl)-6,7,8,9-tetra...)
Affinity DataEC50:  6.06E+3nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317445(7-benzyl-N-neopentyl-5-(piperidin-1-yl)-6,7,8,9-te...)
Affinity DataEC50:  680nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317446(7-benzyl-N-ethyl-5-(piperidin-1-yl)-6,7,8,9-tetrah...)
Affinity DataEC50:  471nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317447(CHEMBL1099135 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  212nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317451(CHEMBL1098838 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  413nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317452(CHEMBL1098837 | N-(7-Benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  433nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317453(CHEMBL1098836 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  63nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317454(CHEMBL1096193 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  99nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317455(CHEMBL1099123 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  123nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317456(CHEMBL1099122 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...)
Affinity DataEC50:  129nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBombesin receptor subtype-3(Rat)
Amri

Curated by ChEMBL
LigandPNGBDBM50317457(7-(4-Fluorobenzoyl)-5-(piperidin-1-yl)-6,7,8,9-tet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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