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Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50031861
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhems-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50035131((+)-(6R,11S)-6,11-dimethyl-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 opioid receptor from guinea pig brain cortex after 150 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhems-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50002051((+/-)-(2RS)-2-[(4RS)-2,2-Diphenyl-1,3-dioxolan-4-y...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 opioid receptor from guinea pig brain cortex after 150 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhems-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM81982(CAS_97-39-2 | DITOLYLGUANIDINE | DTG | Di-o-tolylg...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 opioid receptor from guinea pig brain cortex after 150 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhems-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50320702((+/-)-(2RS)-2-[(4RS)-2,2-Diphenyl-1,3-dioxolan-4-y...)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 opioid receptor from guinea pig brain cortex after 150 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhems-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50320701((+/-)-4-hydroxydioxadrol | CHEMBL1164041)
Affinity DataKi:  971nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 opioid receptor from guinea pig brain cortex after 150 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed