Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50031963
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50322368((S)-5-((S)-1-((S)-2-((S)-1-((S)-1-((S)-1-carboxy-3...)
Affinity DataEC50:  11nMAssay Description:Binding affinity to human NTR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2010
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Rat)
Medical University of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50322368((S)-5-((S)-1-((S)-2-((S)-1-((S)-1-((S)-1-carboxy-3...)
Affinity DataKd:  23nMAssay Description:Displacement of [125I]NT from rat NTR2 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2010
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Medical University of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50322368((S)-5-((S)-1-((S)-2-((S)-1-((S)-1-((S)-1-carboxy-3...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at rat NTR1 expressed in LTK cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2010
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Medical University of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50322368((S)-5-((S)-1-((S)-2-((S)-1-((S)-1-((S)-1-carboxy-3...)
Affinity DataEC50:  54nMAssay Description:Binding affinity to human NTR2 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2010
Entry Details Article
PubMed