Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 3593
TargetTubulin--tyrosine ligase(Human)
Binghamton University

LigandChemical structure of BindingDB Monomer ID 18129BDBM18129((2S)-2-amino-3-(4-hydroxyphenyl)propanoic acid | L...)
Affinity DataKi:  2.50E+4nM ΔG°:  -27.3kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTubulin--tyrosine ligase(Human)
Binghamton University

LigandChemical structure of BindingDB Monomer ID 36555BDBM36555(3-Aminotyrosine)
Affinity DataKi:  2.00E+5nM ΔG°:  -22.0kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2011
Entry Details Article
PubMed
TargetTubulin--tyrosine ligase(Human)
Binghamton University

LigandChemical structure of BindingDB Monomer ID 36556BDBM36556(3-Azidotyrosine)
Affinity DataKi:  2.00E+5nM ΔG°:  -22.0kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2011
Entry Details Article
PubMed
TargetTubulin--tyrosine ligase(Human)
Binghamton University

LigandChemical structure of BindingDB Monomer ID 36557BDBM36557(3-Formyltyrosine)
Affinity DataKi:  3.00E+5nM ΔG°:  -20.9kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2011
Entry Details Article
PubMed
TargetTubulin--tyrosine ligase(Human)
Binghamton University

LigandChemical structure of BindingDB Monomer ID 36554BDBM36554(3-Nitrotyrosine)
Affinity DataKi:  4.00E+5nM ΔG°:  -20.2kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2011
Entry Details Article
PubMed
TargetTubulin--tyrosine ligase(Human)
Binghamton University

LigandChemical structure of BindingDB Monomer ID 36558BDBM36558(4-Aminophenylalanine)
Affinity DataKi: >4.00E+6nM ΔG°: >-14.2kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2011
Entry Details Article
PubMed