Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50032002
Target5-hydroxytryptamine receptor 1A(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Human)
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Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]CCK-8 from human recombinant CCKA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]AB-MECA from human recombinant A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 5A(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323051(1-Biphenyl-3-yl-ethanone, O-(1-naphthylaminocarbon...)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323050(1-Biphenyl-3-yl-ethanone, O-(4-fluorophenylaminoca...)
Affinity DataIC50:  17nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323049(1-Biphenyl-3-yl-ethanone, O-(4-methoxyphenylaminoc...)
Affinity DataIC50:  28nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323052(1-Biphenyl-3-yl-ethanone, O-(phenylaminocarbonyl)o...)
Affinity DataIC50:  69nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323042(1-(3'-Aminocarbonyl-biphenyl-3-yl)-ethanone, O-(ph...)
Affinity DataIC50:  84nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323047(1-Biphenyl-3-yl-ethanone, O-[(4-pentylphenyl)amino...)
Affinity DataIC50:  100nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323043(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(1-piperidi...)
Affinity DataIC50:  112nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323044(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(dodecylami...)
Affinity DataIC50:  116nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323057(1-(4-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323046(1-Biphenyl-3-yl-ethanone, O-(1-piperidinocarbonyl)...)
Affinity DataIC50:  220nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323048(1-Biphenyl-3-yl-ethanone, O-[(5-benzo[b]thiophenyl...)
Affinity DataIC50:  232nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323058(1-Biphenyl-4-yl-ethanone, O-(1-naphthylaminocarbon...)
Affinity DataIC50:  401nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323059(1-Biphenyl-4-yl-ethanone, O-(phenylaminocarbonyl)o...)
Affinity DataIC50:  760nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323056(1-[4-(cyclohexyl)-phenyl]-ethanone,O-(1-naphthylam...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323055(1-[4-(2,5-Dimethyl-pyrrol-1-yl)-phenyl]-ethanone,O...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Mouse)
Università

Curated by ChEMBL
LigandPNGBDBM50323054(1-[2,2']Bithiophenyl-5-yl-ethanone, O-(1-naphthyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP 12177 from human recombinant beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]BRL 43694 from human recombinant 5HT3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1B(Rat)
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Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]CYP from 5HT1B receptor expressed in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]SQ 29548 from human recombinant TXA2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]nociceptin from human recombinant ORL1 receptor expressed in H recombinant HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]U69593 from rat recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeurotensin receptor type 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NT1 receptor expressed in H recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]peptide YY from human recombinant Y2 receptor expressed in KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuropeptide Y receptor type 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]peptide YY from human recombinant Y1 receptor expressed in SK-NM- cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuromedin-K receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]SR 142801 from human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSubstance-K receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]NKA from human recombinant NK2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]4-DAMP from human recombinant muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]AF-DX 384 from human recombinant muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]pirenzepine from human recombinant muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]NDP-a-MSH from human recombinant MC4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistamine H2 receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]APT from human recombinant histamine H2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistamine H1 receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetC-C chemokine receptor type 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]MIP-1a from human recombinant CCR1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetC-X-C chemokine receptor type 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]IL-8 from human recombinant CXCR2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGalanin receptor type 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]Galanin from human recombinant GAL2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]SCH 23390 from human recombinant dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetB2 bradykinin receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]bradykinin from human recombinant bradykinin B2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetType-1 angiotensin II receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I][Sar1,Ile8]-AT II from human recombinant AT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP 12177 from human recombinant beta-1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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