Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50032006
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323107((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(pyridin-4-y...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323100((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(1-(2-(4-met...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323106((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(1-(2-morpho...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323113((R)-5-(5-(pyridin-4-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323105((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(2-(1-methyl...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323116((R)-5-(5-(pyridin-3-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323102((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(1-(3-(4-eth...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323122((R)-5-(5-(1-methyl-1H-pyrazol-4-yl)-1H-benzo[d]imi...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323121((R)-5-(5-(1H-pyrazol-4-yl)-1H-benzo[d]imidazol-1-y...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323124((R)-5-(5-(2-methylpyridin-4-yl)-1H-benzo[d]imidazo...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323123((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(6-(1-methyl-1H...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323109((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(1-methyl-1H...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323110((R)-5-(5-(2-aminopyrimidin-4-yl)-1H-benzo[d]imidaz...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323108((R)-5-(5-(2-aminopyridin-4-yl)-1H-benzo[d]imidazol...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323127((R)-5-(5-(2-aminopyrimidin-5-yl)-1H-benzo[d]imidaz...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323098((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(2-(1-methyl...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323097((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(2-(2-hydrox...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323096((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(2-(2-(methy...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323114((R)-5-(6-(pyridin-4-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323099((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(6-(1-methyl...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323117((R)-5-(6-(pyridin-3-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323115((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(6-(pyridin-4-y...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323101((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(1-(3-(dimet...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323104((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(2-(4-methyl...)
Affinity DataIC50: 2nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323093((R)-5-(5-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323119((R)-5-(5-(thiophen-2-yl)-1H-benzo[d]imidazol-1-yl)...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323095((R)-5-(5-(2-(2-(dimethylamino)ethylamino)pyridin-4...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323125((R)-5-(5-(2-chloropyridin-4-yl)-1H-benzo[d]imidazo...)
Affinity DataIC50: 4nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323110((R)-5-(5-(2-aminopyrimidin-4-yl)-1H-benzo[d]imidaz...)
Affinity DataIC50: 5nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323094((R)-5-(5-(2-morpholinopyridin-4-yl)-1H-benzo[d]imi...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323120((R)-5-(5-(1H-pyrrol-2-yl)-1H-benzo[d]imidazol-1-yl...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323122((R)-5-(5-(1-methyl-1H-pyrazol-4-yl)-1H-benzo[d]imi...)
Affinity DataIC50: 6nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323118((R)-5-(5-(pyridin-2-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323109((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(1-methyl-1H...)
Affinity DataIC50: 6nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323111((R)-5-(5-phenyl-1H-benzo[d]imidazol-1-yl)-3-(1-(2-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323113((R)-5-(5-(pyridin-4-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323103((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(2-(piperazi...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323107((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(pyridin-4-y...)
Affinity DataIC50: 10nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323123((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(6-(1-methyl-1H...)
Affinity DataIC50: 13nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323114((R)-5-(6-(pyridin-4-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323116((R)-5-(5-(pyridin-3-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323112((R)-5-(6-phenyl-1H-benzo[d]imidazol-1-yl)-3-(1-(2-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323115((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(6-(pyridin-4-y...)
Affinity DataIC50: 25nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323117((R)-5-(6-(pyridin-3-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323119((R)-5-(5-(thiophen-2-yl)-1H-benzo[d]imidazol-1-yl)...)
Affinity DataIC50: 50nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323126((R)-5-(6-(2-chloropyridin-4-yl)-1H-benzo[d]imidazo...)
Affinity DataIC50: 53nMAssay Description:Inhibition of PLK1 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323118((R)-5-(5-(pyridin-2-yl)-1H-benzo[d]imidazol-1-yl)-...)
Affinity DataIC50: 79nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323094((R)-5-(5-(2-morpholinopyridin-4-yl)-1H-benzo[d]imi...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant CYP2C9 using 7-methoxy-4-trifluoromethylcoumarin-3-acetic acid as substrate by fluorescence plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323107((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(5-(pyridin-4-y...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant CYP2C9 using 7-{3-(4-phenylpiperazin-1-ylmethyl)benzyl}resorufin as substrate by fluorescence plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50323120((R)-5-(5-(1H-pyrrol-2-yl)-1H-benzo[d]imidazol-1-yl...)
Affinity DataIC50: 126nMAssay Description:Inhibition of full lungth PLK3 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
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