Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50022509
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM50380387(CHEMBL2018451)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM50261816(tert-butyl 4-(3-((7-(hydroxyamino)-7-oxoheptyl)car...)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM22449(N-(4-{(2R,4R,6S)-4-{[(4,5-diphenyl-1,3-oxazol-2-yl...)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124194(US8748451, 10)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124190(US8748451, 5)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM50331109(CHEMBL1290142 | US8748451, 1 | 6-(9H-carbazol-9-yl...)
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124187(US8748451, 2)
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124196(US8748451, 12)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124189(US8748451, 4)
Affinity DataIC50: 213nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124195(US8748451, 11)
Affinity DataIC50: 301nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124188(US8748451, 7 | US8748451, 3)
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124192(US8748451, 8)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124193(US8748451, 9)
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHistone deacetylase 6(Human)TBA
LigandPNGBDBM124197(US8748451, 13)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic RHKKAc peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed