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Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50032072
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323914(CHEMBL1213786 | Tamoxifen butyl bromide)
Affinity DataKi:  13.0nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323912(CHEMBL1213784 | Tamoxifen ethyl bromide)
Affinity DataKi:  13.7nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323913(CHEMBL1213785 | Tamoxifen isopropyl bromide)
Affinity DataKi:  25.4nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataKi:  31.2nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323911(CHEMBL1213783 | Tamoxifen methyl iodide)
Affinity DataKi:  46.3nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed