Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50032079
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM20880((2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)me...)
Affinity DataIC50:  0.490nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324016((2R,3R,4S,5S,6R)-2-(5-Chloro-4-(4-ethylbenzyl)thia...)
Affinity DataIC50:  121nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324017((2R,3R,4S,5S,6R)-2-(4-(4-Butylbenzyl)-5-chlorothia...)
Affinity DataIC50:  251nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324015((2R,3R,4S,5S,6R)-2-(4-Chloro-5-(4-methylbenzyl)thi...)
Affinity DataIC50:  257nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324018((2R,3R,4S,5S,6R)-2-(4-(Biphenyl-4-ylmethyl)-5-chlo...)
Affinity DataIC50:  411nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324002((2S,3R,4R,5S,6R)-2-(6-chloro-5-(4-methoxybenzyl)py...)
Affinity DataIC50:  610nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324012((2R,3R,4S,5S,6R)-2-(4-Bromo-5-(4-ethylbenzyl)thiaz...)
Affinity DataIC50:  786nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324011((2R,3R,4S,5S,6R)-2-(4-Bromo-5-(4-methylbenzyl)thia...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324013((2R,3R,4S,5S,6R)-2-(4-Bromo-5-(4-tert-butylbenzyl)...)
Affinity DataIC50:  2.36E+3nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324004((2R,3S,4S,5R,6R)-2-(Hydroxymethyl)-6-(5-(4-methylb...)
Affinity DataIC50:  4.63E+3nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324014((2R,3R,4S,5S,6R)-2-(4-Bromo-5-(4-chlorobenzyl)thia...)
Affinity DataIC50:  8.64E+3nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324006((2R,3R,4S,5S,6R)-2-(5-(4-tert-Butylbenzyl)thiazol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324007((2R,3S,4S,5R,6R)-2-(Hydroxymethyl)-6-(4-(4-methylb...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324009((2R,3S,4S,5R,6R)-2-(Hydroxymethyl)-6-(4-(4-propylb...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324005((2R,3R,4S,5S,6R)-2-(5-(4-Chlorobenzyl)thiazol-2-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324010((2R,3R,4S,5S,6R)-2-(5-Benzyl-4-bromothiazol-2-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324003((2R,3R,4S,5S,6R)-2-(5-Benzylthiazol-2-yl)-6-(hydro...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50324008((2R,3R,4S,5S,6R)-2-(4-(4-Ethylbenzyl)thiazol-2-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed