Compile Data Set for Download or QSAR
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Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50032300
TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326858(CHEMBL1254556 | N-((3R,4R,5S,6R)-2,4-bis(4-chlorob...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326859(CHEMBL1254630 | N-((3R,4R,5S,6R)-4-(4-chlorobenzyl...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326860(CHEMBL1254711 | N-((3R,4R,5S,6R)-2-(4-chlorobenzyl...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326861(CHEMBL1254796 | N-((3R,4R,5S,6R)-4-(4-chlorobenzyl...)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326862(4-(diaminomethyleneamino)-N-((3R,4R,5S,6R)-5-hydro...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326863(3-(diaminomethyleneamino)-N-((3R,4R,5S,6R)-5-hydro...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326864(CHEMBL1254883 | N-((3R,4R,5S,6R)-4-(4-chlorobenzyl...)
Affinity DataKi:  6.60E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326854((Naphth-2-yl)methyl-2-(4'-Aminobutyrylamido)-3-O-(...)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326878((2R,3S,5R)-5-(3-aminopropylamino)-4-(4-chlorobenzy...)
Affinity DataIC50:  70nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326872(CHEMBL1254140 | Naphth-2-yl)methyl-2-(4'-Aminobuty...)
Affinity DataIC50:  70nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326879((2R,3S,5R)-5-(2-aminoethylamino)-2-(methoxymethyl)...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326865((4'-Chlorobenzyl)3-O-(4'-Chlorobenzyl)-2-deoxy-2-(...)
Affinity DataIC50:  120nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326881((2R,3S,5R)-5-(2-aminoethylamino)-2-(methoxymethyl)...)
Affinity DataIC50:  160nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326880((2R,3S,5R)-5-(2-aminoethylamino)-4-(benzyloxy)-2-(...)
Affinity DataIC50:  160nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326874(CHEMBL1254882 | N-((2S,3R,4S,5S,6R)-6-(benzyloxyme...)
Affinity DataIC50:  180nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326856(4-amino-N-((2R,3R,4R,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50:  180nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326857((Naphth-2-yl)methyl-2-(3'-Aminopropionylamido)-2-d...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326855(4-amino-N-((2S,3R,4S,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326882((2R,3S,5R)-5-(3-aminopropylamino)-2-(methoxymethyl...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 3(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326857((Naphth-2-yl)methyl-2-(3'-Aminopropionylamido)-2-d...)
Affinity DataIC50:  380nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326873(3-amino-N-((2S,3R,4S,5S,6R)-6-((4-chlorobenzyloxy)...)
Affinity DataIC50:  430nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 3(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326854((Naphth-2-yl)methyl-2-(4'-Aminobutyrylamido)-3-O-(...)
Affinity DataIC50:  430nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326875(3-amino-N-((2S,3R,4S,5S,6R)-5-hydroxy-2-(methylthi...)
Affinity DataIC50:  440nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326869(4'-Chlorobenzyl-2-Deoxy-2-(4'-guanidinobutyrylamid...)
Affinity DataIC50:  450nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 3(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326872(CHEMBL1254140 | Naphth-2-yl)methyl-2-(4'-Aminobuty...)
Affinity DataIC50:  500nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326870(2'-(Phenyl)ethyl-3-O-(4'-Chlorobenzyl)-2-deoxy-2-(...)
Affinity DataIC50:  540nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 2(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326857((Naphth-2-yl)methyl-2-(3'-Aminopropionylamido)-2-d...)
Affinity DataIC50:  650nMAssay Description:Displacement of [125I]iodotyrosyl from human SST2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326876(3-amino-N-((2S,3R,4S,5S,6R)-6-(benzyloxymethyl)-5-...)
Affinity DataIC50:  660nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326877(CHEMBL1253871 | N-((2S,3R,4S,5S,6R)-6-((4-chlorobe...)
Affinity DataIC50:  720nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326867((Naphth-2-yl)methyl-3-O-(4'-Chlorobenzyl)-2-deoxy-...)
Affinity DataIC50:  920nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 2(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326873(3-amino-N-((2S,3R,4S,5S,6R)-6-((4-chlorobenzyloxy)...)
Affinity DataIC50:  980nMAssay Description:Displacement of [125I]iodotyrosyl from human SST2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326871((Naphth-2-yl)methyl-2-Deoxy-2-(4'-guanidinobutyryl...)
Affinity DataIC50:  1.16E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 3(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326856(4-amino-N-((2R,3R,4R,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50:  1.32E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326866((4'-Chlorobenzyl)3-O-(4'-Chlorobenzyl)-2-deoxy-2-(...)
Affinity DataIC50:  1.66E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanin-concentrating hormone receptor 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326868((Naphth-2-yl)methyl-3-O-(4'-Chlorobenzyl)-2-deoxy-...)
Affinity DataIC50:  1.75E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326857((Naphth-2-yl)methyl-2-(3'-Aminopropionylamido)-2-d...)
Affinity DataIC50:  2.80E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 2(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326856(4-amino-N-((2R,3R,4R,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50:  3.32E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326857((Naphth-2-yl)methyl-2-(3'-Aminopropionylamido)-2-d...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 5(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326873(3-amino-N-((2S,3R,4S,5S,6R)-6-((4-chlorobenzyloxy)...)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 2(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326855(4-amino-N-((2S,3R,4S,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50:  6.10E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 3(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326873(3-amino-N-((2S,3R,4S,5S,6R)-6-((4-chlorobenzyloxy)...)
Affinity DataIC50:  6.33E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 3(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326855(4-amino-N-((2S,3R,4S,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50:  8.40E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326873(3-amino-N-((2S,3R,4S,5S,6R)-6-((4-chlorobenzyloxy)...)
Affinity DataIC50:  9.59E+3nMAssay Description:Displacement of [125I]iodotyrosyl from human SST1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 2(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326872(CHEMBL1254140 | Naphth-2-yl)methyl-2-(4'-Aminobuty...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326855(4-amino-N-((2S,3R,4S,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326854((Naphth-2-yl)methyl-2-(4'-Aminobutyrylamido)-3-O-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326856(4-amino-N-((2R,3R,4R,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326855(4-amino-N-((2S,3R,4S,5S,6R)-5-hydroxy-6-(methoxyme...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 4(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326854((Naphth-2-yl)methyl-2-(4'-Aminobutyrylamido)-3-O-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSomatostatin receptor type 1(Human)
Alchemia

Curated by ChEMBL
LigandPNGBDBM50326872(CHEMBL1254140 | Naphth-2-yl)methyl-2-(4'-Aminobuty...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]iodotyrosyl from human SST1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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